A CONVENIENT SYNTHESIS OF 2-AMINO-6-METHOXY-1-METHYLCARBAZOLE AND 2-AMINO-6-METHOXY-1,4-DIMETHYLCARBAZOLE DERIVATIVES AND THEIR 6-AZA ANALOGS

被引：8

作者：

MORON, J

LANDRAS, C

BISAGNI, E

机构：

[1] URA 1387 CNRS, Institut Curie, Section de Biologie, Centre Universitaire, Orsay, F-91405

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1992年 / 29卷 / 06期

关键词：

D O I：

10.1002/jhet.5570290634

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2,6-Diaminotoluene (3a) and 2,6-diamino-p-xylene (3c) led to 2-methyl (and 2,5-dimethyl)-3-acetylamino-phenylhydrazines 5a,b. Fischer indolization of their hydrazones 6a,b and 7a,b derived from 4-methoxycyclohexanone and 4-piperidone, and subsequent aromatization of intermediate tetrahydrocarbazole derivatives 8a,b and 9a,b allowed us to work out a convenient route to the title compounds.

引用

页码：1573 / 1576

页数：4

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