ACUTE STRESS INDUCES AN INCREASE IN RAT CEREBRAL-CORTEX LEVELS OF NORMAL-BUTYL-BETA-CARBOLINE-3-CARBOXYLATE, AN ENDOGENOUS BENZODIAZEPINE BINDING INHIBITOR

被引:23
作者
MEDINA, JH [1 ]
PENA, C [1 ]
NOVAS, ML [1 ]
PALADINI, AC [1 ]
DEROBERTIS, E [1 ]
机构
[1] UNIV BUENOS AIRES,CONSEJO NACL INVEST CIENT & TECN,FAC FARM & BIOQUIM,RA-1113 BUENOS AIRES,ARGENTINA
关键词
D O I
10.1016/0197-0186(87)90043-X
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:255 / 259
页数:5
相关论文
共 17 条
[1]   BENZODIAZEPINE RECEPTORS IN THE BRAIN AS AFFECTED BY DIFFERENT EXPERIMENTAL STRESSES - CHANGES ARE SMALL AND NOT UNDIRECTIONAL [J].
BRAESTRUP, C ;
NIELSEN, M ;
NIELSEN, EB ;
LYON, M .
PSYCHOPHARMACOLOGY, 1979, 65 (03) :273-277
[2]   URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M ;
OLSEN, CE .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2288-2292
[3]   SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].
BRAESTRUP, C ;
SQUIRES, RF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809
[4]  
DEBLAS AL, 1986, SOC NEUR ABSTR, V53, P185
[5]   CHOLINERGIC MUSCARINIC RECEPTORS IN RAT CEREBRAL-CORTEX, BASAL GANGLIA AND CEREBELLUM UNDERGO RAPID AND REVERSIBLE CHANGES AFTER ACUTE STRESS [J].
ESTEVEZ, EE ;
JERUSALINSKY, D ;
MEDINA, JH ;
DEROBERTIS, E .
NEUROSCIENCE, 1984, 13 (04) :1353-1357
[6]   A BRAIN OCTADECANEUROPEPTIDE GENERATED BY TRYPTIC DIGESTION OF DBI (DIAZEPAM BINDING INHIBITOR) FUNCTIONS AS A PROCONFLICT LIGAND OF BENZODIAZEPINE RECOGNITION SITES [J].
FERRERO, P ;
GUIDOTTI, A ;
CONTITRONCONI, B ;
COSTA, E .
NEUROPHARMACOLOGY, 1984, 23 (11) :1359-1362
[7]   BENZODIAZEPINES REDUCE STRESS-AUGMENTED INCREASE IN RAT URINE MONOAMINE-OXIDASE INHIBITOR [J].
GLOVER, V ;
BHATTACHARYA, SK ;
SANDLER, M ;
FILE, SE .
NATURE, 1981, 292 (5821) :347-349
[8]   ISOLATION, CHARACTERIZATION, AND PURIFICATION TO HOMOGENEITY OF AN ENDOGENOUS POLYPEPTIDE WITH AGONISTIC ACTION ON BENZODIAZEPINE RECEPTORS [J].
GUIDOTTI, A ;
FORCHETTI, CM ;
CORDA, MG ;
KONKEL, D ;
BENNETT, CD ;
COSTA, E .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (11) :3531-3535
[9]   SEARCHING FOR ENDOGENOUS LIGAND(S) OF CENTRAL BENZODIAZEPINE RECEPTORS [J].
HAMON, M ;
SOUBRIE, P .
NEUROCHEMISTRY INTERNATIONAL, 1983, 5 (06) :663-672
[10]  
KORNEYEV AY, 1983, MOL PHARMACOL, V23, P310