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METHODS FOR DRUG DISCOVERY - DEVELOPMENT OF POTENT, SELECTIVE, ORALLY EFFECTIVE CHOLECYSTOKININ ANTAGONISTS
被引:1316
作者
:
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
EVANS, BE
[
1
]
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
RITTLE, KE
[
1
]
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
BOCK, MG
[
1
]
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
DIPARDO, RM
[
1
]
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
FREIDINGER, RM
[
1
]
WHITTER, WL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
WHITTER, WL
[
1
]
LUNDELL, GF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
LUNDELL, GF
[
1
]
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
VEBER, DF
[
1
]
ANDERSON, PS
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
ANDERSON, PS
[
1
]
CHANG, RSL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
CHANG, RSL
[
1
]
LOTTI, VJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
LOTTI, VJ
[
1
]
CERINO, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
CERINO, DJ
[
1
]
CHEN, TB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
CHEN, TB
[
1
]
KLING, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
KLING, PJ
[
1
]
KUNKEL, KA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
KUNKEL, KA
[
1
]
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
SPRINGER, JP
[
1
]
HIRSHFIELD, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
HIRSHFIELD, J
[
1
]
机构
:
[1]
MERCK INST THERAPEUT RES,RAHWAY,NJ 07065
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1988年
/ 31卷
/ 12期
关键词
:
D O I
:
10.1021/jm00120a002
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:2235 / 2246
页数:12
相关论文
共 56 条
[1]
DIAZEPAM-BINDING INHIBITOR - A NEUROPEPTIDE LOCATED IN SELECTED NEURONAL POPULATIONS OF RAT-BRAIN
ALHO, H
论文数:
0
引用数:
0
h-index:
0
ALHO, H
COSTA, E
论文数:
0
引用数:
0
h-index:
0
COSTA, E
FERRERO, P
论文数:
0
引用数:
0
h-index:
0
FERRERO, P
FUJIMOTO, M
论文数:
0
引用数:
0
h-index:
0
FUJIMOTO, M
COSENZAMURPHY, D
论文数:
0
引用数:
0
h-index:
0
COSENZAMURPHY, D
GUIDOTTI, A
论文数:
0
引用数:
0
h-index:
0
GUIDOTTI, A
[J].
SCIENCE,
1985,
229
(4709)
: 179
-
182
[2]
THE CHOLECYSTOKININ ANTAGONIST L-364,718 INHIBITS THE ACTION OF CHOLECYSTOKININ BUT NOT BOMBESIN ON RAT PANCREATIC-SECRETION INVIVO
ANDERSON, L
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
ANDERSON, L
DOCKRAY, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
DOCKRAY, GJ
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1988,
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311
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ARIENS EJ, 1979, RECEPTORS COMPREHENS, V1, P33
[4]
A REARRANGEMENT OF 5-ARYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPINE-2-14-OXIDES
BELL, SC
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0
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0
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0
BELL, SC
CHILDRESS, SJ
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0
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0
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0
CHILDRESS, SJ
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1962,
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BELL SC, 1964, J HETEROCYCL CHEM, V4, P647
[6]
BELL SC, 1965, Patent No. 3198789
[7]
BLOUNT JF, 1983, MOL PHARM, V24, P426
[8]
AN EXPEDIENT SYNTHESIS OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONE
BOCK, MG
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0
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h-index:
0
BOCK, MG
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
FREIDINGER, RM
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0
引用数:
0
h-index:
0
FREIDINGER, RM
[J].
TETRAHEDRON LETTERS,
1987,
28
(09)
: 939
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942
[9]
SYNTHESIS AND RESOLUTION OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONES
BOCK, MG
论文数:
0
引用数:
0
h-index:
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机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
BOCK, MG
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
DIPARDO, RM
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
EVANS, BE
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
RITTLE, KE
VEBER, DF
论文数:
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h-index:
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机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
VEBER, DF
FREIDINGER, RM
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MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
FREIDINGER, RM
HIRSHFIELD, J
论文数:
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引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
HIRSHFIELD, J
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
SPRINGER, JP
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1987,
52
(15)
: 3232
-
3239
[10]
BENZODIAZEPINES ANTAGONIZE CHOLECYSTOKININ-INDUCED ACTIVATION OF RAT HIPPOCAMPAL-NEURONS
BRADWEJN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
BRADWEJN, J
DEMONTIGNY, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
DEMONTIGNY, C
[J].
NATURE,
1984,
312
(5992)
: 363
-
364
←
1
2
3
4
5
6
→
共 56 条
[1]
DIAZEPAM-BINDING INHIBITOR - A NEUROPEPTIDE LOCATED IN SELECTED NEURONAL POPULATIONS OF RAT-BRAIN
ALHO, H
论文数:
0
引用数:
0
h-index:
0
ALHO, H
COSTA, E
论文数:
0
引用数:
0
h-index:
0
COSTA, E
FERRERO, P
论文数:
0
引用数:
0
h-index:
0
FERRERO, P
FUJIMOTO, M
论文数:
0
引用数:
0
h-index:
0
FUJIMOTO, M
COSENZAMURPHY, D
论文数:
0
引用数:
0
h-index:
0
COSENZAMURPHY, D
GUIDOTTI, A
论文数:
0
引用数:
0
h-index:
0
GUIDOTTI, A
[J].
SCIENCE,
1985,
229
(4709)
: 179
-
182
[2]
THE CHOLECYSTOKININ ANTAGONIST L-364,718 INHIBITS THE ACTION OF CHOLECYSTOKININ BUT NOT BOMBESIN ON RAT PANCREATIC-SECRETION INVIVO
ANDERSON, L
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
ANDERSON, L
DOCKRAY, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
UNIV LIVERPOOL,PHYSIOL LAB,MRC,SECRETORY CONTROL GRP,POB 147,LIVERPOOL L69 3BX,ENGLAND
DOCKRAY, GJ
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1988,
146
(2-3)
: 307
-
311
[3]
ARIENS EJ, 1979, RECEPTORS COMPREHENS, V1, P33
[4]
A REARRANGEMENT OF 5-ARYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPINE-2-14-OXIDES
BELL, SC
论文数:
0
引用数:
0
h-index:
0
BELL, SC
CHILDRESS, SJ
论文数:
0
引用数:
0
h-index:
0
CHILDRESS, SJ
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1962,
27
(05)
: 1691
-
&
[5]
BELL SC, 1964, J HETEROCYCL CHEM, V4, P647
[6]
BELL SC, 1965, Patent No. 3198789
[7]
BLOUNT JF, 1983, MOL PHARM, V24, P426
[8]
AN EXPEDIENT SYNTHESIS OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONE
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
BOCK, MG
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
DIPARDO, RM
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
EVANS, BE
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
RITTLE, KE
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
VEBER, DF
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
FREIDINGER, RM
[J].
TETRAHEDRON LETTERS,
1987,
28
(09)
: 939
-
942
[9]
SYNTHESIS AND RESOLUTION OF 3-AMINO-1,3-DIHYDRO-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONES
BOCK, MG
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
BOCK, MG
DIPARDO, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
DIPARDO, RM
EVANS, BE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
EVANS, BE
RITTLE, KE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
RITTLE, KE
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
VEBER, DF
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
FREIDINGER, RM
HIRSHFIELD, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
HIRSHFIELD, J
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
SPRINGER, JP
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1987,
52
(15)
: 3232
-
3239
[10]
BENZODIAZEPINES ANTAGONIZE CHOLECYSTOKININ-INDUCED ACTIVATION OF RAT HIPPOCAMPAL-NEURONS
BRADWEJN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
BRADWEJN, J
DEMONTIGNY, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
UNIV MONTREAL,NEUROSCI RES CTR,MONTREAL H3C 3J7,QUEBEC,CANADA
DEMONTIGNY, C
[J].
NATURE,
1984,
312
(5992)
: 363
-
364
←
1
2
3
4
5
6
→