A NOVEL ACCESS TO 4-FLUOROPYRIMIDINES FROM ALPHA-CHLORO-ALPHA'-TRIFLUOROMETHYLKETONES

被引：8

作者：

DENANTEUIL, G

机构：

[1] Institut de Recherches Servier., 11, rue des Moulineaux.

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 22期

关键词：

ALPHA-CHLORO-BETA'-TRIFLUOROMETHYLKETONES; ALPHA-CHLORO-ALPHA'-TRIFLUOROMETHYLKETONES; FORMAMIDINE; 4-FLUOROPYRIMIDINES; TRIFLUOROMETHYL GROUP FLUORINES DISPLACEMENT;

D O I：

10.1016/S0040-4039(00)74355-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

When treated with formamidine acetate and KOH, a-chloro-a'-trifluoromethyl ketones afford, through in moderate yield, 4-fluoropyrimidine derivatives.

引用

页码：2467 / 2468

页数：2

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