UNCONVENTIONAL NUCLEOTIDE ANALOGUES .2. SYNTHESIS OF ADENYL ANALOGUE OF WILLARDIINE

被引：27

作者：

NOLLET, AJH

PANDIT, UK

机构：

[1] Laboratory of Organic Chemistry, University of Amsterdam, Amsterdam

来源：

TETRAHEDRON | 1969年 / 25卷 / 24期

关键词：

D O I：

10.1016/S0040-4020(01)83105-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The Michael addition of adenine (6a), 6-chloropurine (6b) and 2,6-dichloropurine (6c) to methyl α-chloroacrylate gives high yields of the corresponding adducts (7a-7c). Hydrolysis and amination of 7a gave the adenyl analogue of Willardiine (2). © 1969.

引用

页码：5983 / &

共 24 条

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