EFFECTS OF EQUILIBRATION TIME ON THE ATTAINMENT OF EQUILIBRIUM BETWEEN ANTAGONISTS AND DRUG RECEPTORS

被引:41
作者
KENAKIN, TP [1 ]
机构
[1] BURROUGHS WELLCOME CO, WELLCOME RES LABS, DEPT PHARMACOL, 3030 CORNWALLIS RD, RES TRIANGLE PK, NC 27709 USA
关键词
D O I
10.1016/0014-2999(80)90462-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:295 / 306
页数:12
相关论文
共 21 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]  
CHAHL LORIS A., 1967, EUR J PHARMACOL, V2, P77, DOI 10.1016/0014-2999(67)90028-3
[3]   RECEPTOR MECHANISMS [J].
FURCHGOTT, RF .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1964, 4 :21-+
[4]  
FURCHGOTT RF, 1955, PHARMACOL REV, V7, P183
[5]  
Furchgott RF, 1972, HDB EXPT PHARM, V3, P283
[6]  
FURCHGOTT RF, 1973, FRONTIERS CATECHOLAM, P295
[7]   STABILITY OF NORADRENALINE IN PHYSIOLOGICAL SALINE SOLUTIONS [J].
HUGHES, IE ;
SMITH, JA .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1978, 30 (02) :124-126
[8]  
KENAKIN TP, 1978, MOL PHARMACOL, V14, P607
[9]   SOME CHEMICAL AND PHYSICAL PROPERTIES ASSOCIATED WITH HISTAMINE ANTAGONISM [J].
MARSHALL, PB .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1955, 10 (03) :270-278
[10]  
MORAN NC, 1972, FRONTIERS CATECHOLAM, P291