NALOXAZONE IRREVERSIBLY INHIBITS THE HIGH-AFFINITY BINDING OF [I-125]D-ALA2-D-LEU5-ENKEPHALIN

被引:43
作者
HAZUM, E [1 ]
CHANG, KJ [1 ]
CUATRECASAS, P [1 ]
PASTERNAK, GW [1 ]
机构
[1] MEM SLOAN KETTERING CANC CTR,GEORGE C COTZIAS LAB NEURO-ONCOL,NEW YORK,NY 10021
关键词
D O I
10.1016/0024-3205(81)90274-5
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2973 / 2979
页数:7
相关论文
共 14 条
[1]   POSSIBLE ROLE OF DISTINCT MORPHINE AND ENKEPHALIN RECEPTORS IN MEDIATING ACTIONS OF BENZOMORPHAN DRUGS (PUTATIVE-KAPPA AND SIGMA-AGONISTS) [J].
CHANG, KJ ;
HAZUM, E ;
CUATRECASAS, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (08) :4469-4473
[2]  
CHANG KJ, 1978, MOL PHARMACOL, V14, P961
[3]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[4]  
CHANG KJ, 1979, MOL PHARMACOL, V16, P91
[5]  
CHILDERS SR, EUROP J PHARMACOL
[6]   ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].
LORD, JAH ;
WATERFIELD, AA ;
HUGHES, J ;
KOSTERLITZ, HW .
NATURE, 1977, 267 (5611) :495-499
[7]   OPIATE ANALGESIA - EVIDENCE FOR MEDIATION BY A SUB-POPULATION OF OPIATE RECEPTORS [J].
PASTERNAK, GW ;
CHILDERS, SR ;
SNYDER, SH .
SCIENCE, 1980, 208 (4443) :514-516
[8]   IDENTIFICATION OF NOVEL HIGH AFFINITY OPIATE RECEPTOR-BINDING IN RAT-BRAIN [J].
PASTERNAK, GW ;
SNYDER, SH .
NATURE, 1975, 253 (5492) :563-565
[9]   MULTIPLE OPIATE RECEPTORS - [H-3]ETHYLKETOCYCLAZOCINE RECEPTOR-BINDING AND KETOCYCLAZOCINE ANALGESIA [J].
PASTERNAK, GW .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (06) :3691-3694
[10]  
PASTERNAK GW, 1980, J PHARMACOL EXP THER, V214, P455