PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .13. POTENTIAL IRREVERSIBLE NARCOTIC ANTAGONIST-BASED LIGANDS DERIVED FROM 6,14-ENDO-ETHENOTETRAHYDROORIPAVINE WITH 7-(METHOXYFUMAROYL)AMINO, (BROMOACETYL)AMINO, OR ISOTHIOCYANATE ELECTROPHILES - CHEMISTRY, BIOCHEMISTRY, AND PHARMACOLOGYV

被引：13

作者：

LESSOR, RA

BAJWA, BS

RICE, KC

JACOBSON, AE

STREATY, RA

KLEE, WA

SMITH, CB

ACETO, MD

MAY, EL

HARRIS, LS

机构：

[1] NIDDKD, CHEM LAB, MED CHEM SECT, BETHESDA, MD 20892 USA

[2] NIMH, GEN & COMPARAT BIOCHEM LAB, BETHESDA, MD 20892 USA

[3] UNIV MICHIGAN, DEPT PHARMACOL, ANN ARBOR, MI 48109 USA

[4] VIRGINIA COMMONWEALTH UNIV, MED COLL VIRGINIA, DEPT PHARMACOL, RICHMOND, VA 23298 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 11期

关键词：

D O I：

10.1021/jm00161a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2136 / 2141

页数：6

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