AN EFFICIENT ROUTE TO C-4 LINKED IMIDAZOLE NUCLEOSIDES - SYNTHESIS OF 2-CARBAMOYL-4-(2'-DEOXY-BETA-D-RIBOFURANOSYL)IMIDAZOLE

被引：24

作者：

BERGSTROM, DE ^{[1
]}

ZHANG, PM ^{[1
]}

机构：

[1] WALTHER CANC INST,INDIANAPOLIS,IN 46208

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 45期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/0040-4039(91)80199-G

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The first synthesis of an imidazole C-nucleoside linked through C-4, 2-carbamoyl-4-(2'-deoxy-beta-D-ribofuranosyl) imidazole was achieved by way of a nine-step sequence starting from 2-deoxy-3, 5-di-O-p-toluoyl-D-erythro-pentofuranosyl chloride.

引用

页码：6485 / 6488

页数：4

共 16 条

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