DRUGS FROM EMASCULATED HORMONES - THE PRINCIPLE OF SYNTOPIC ANTAGONISM (NOBEL LECTURE)

被引:14
作者
BLACK, JW
机构
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D O I
10.1002/anie.198908861
中图分类号
O6 [化学];
学科分类号
0703 ;
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页码:886 / 894
页数:9
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共 35 条
[1]   A STUDY OF THE ADRENOTROPIC RECEPTORS [J].
AHLQUIST, RP .
AMERICAN JOURNAL OF PHYSIOLOGY, 1948, 153 (03) :586-600
[2]  
ARIENS EJ, 1954, ARCH INT PHARMACOD T, V99, P32
[3]   RECEPTORS MEDIATING SOME ACTIONS OF HISTAMINE [J].
ASH, ASF ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1966, 27 (02) :427-&
[4]   ANTAGONISM OF AN INDIRECTLY ACTING AGONIST - BLOCK BY PROPRANOLOL AND SOTALOL OF THE ACTION OF TYRAMINE ON RAT-HEART [J].
BLACK, JW ;
JENKINSON, DH ;
KENAKIN, TP .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 65 (01) :1-10
[5]   OPERATIONAL MODELS OF PHARMACOLOGICAL AGONISM [J].
BLACK, JW ;
LEFF, P .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1983, 220 (1219) :141-162
[6]   THE EFFECTS OF 5-HYDROXYTRYPTAMINE ON GASTRIC SECRETION IN ANAESTHETIZED DOGS [J].
BLACK, JW ;
FISHER, EW ;
SMITH, AN .
JOURNAL OF PHYSIOLOGY-LONDON, 1958, 141 (01) :27-34
[7]   AN OPERATIONAL MODEL OF PHARMACOLOGICAL AGONISM - THE EFFECT OF E/[A] CURVE SHAPE ON AGONIST DISSOCIATION-CONSTANT ESTIMATION [J].
BLACK, JW ;
LEFF, P ;
SHANKLEY, NP ;
WOOD, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (02) :561-571
[8]   PHARMACOLOGICAL ANALYSIS OF THE PENTAGASTRIN-TIOTIDINE INTERACTION IN THE MOUSE ISOLATED STOMACH [J].
BLACK, JW ;
LEFF, P ;
SHANKLEY, NP .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 86 (03) :589-599
[9]  
BLACK JW, 1964, LANCET, V1, P1081
[10]  
BLACK JW, 1962, LANCET, V2, P311