SYNTHESIS OF MEDIUM RING LACTAMS VIA CYCLIZATION REACTIONS USING POLYMER-BOUND HOBT AS CATALYST

被引：28

作者：

HUANG, W ^{[1
]}

KALIVRETENOS, AG ^{[1
]}

机构：

[1] UNIV MARYLAND BALTIMORE CTY,DEPT CHEM & BIOCHEM,BALTIMORE,MD 21228

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 50期

关键词：

D O I：

10.1016/0040-4039(95)01977-P

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of medium ring lactams (7-, 9-, 11- and 13-membered rings) via cyclization reactions mediated by polymer bound 1-hydroxybenzotriazole (HOBT) is reported.

引用

页码：9113 / 9116

页数：4

共 17 条

[1]

BECKMANN E, 1986, CHEM BER, V89, P988

[2]

Cawley R. E, 1987, ORG REACTIONS, V35, P1

[3] CENTRAL NERVOUS-SYSTEM ACTIVE COMPOUNDS .2. SYNTHESIS OF SOME 4-SUBSTITUTED, 5-SUBSTITUTED, 6-SUBSTITUTED AND 7-SUBSTITUTED CAPROLACTAMS [J].

DUONG, T ;

PRAGER, RH ;

TIPPETT, JM ;

WARD, AD ;

KERR, DIB .

AUSTRALIAN JOURNAL OF CHEMISTRY, 1976, 29 (12) :2667-2682

[4] CNS ACTIVITIES OF LACTAM DERIVATIVES [J].

ELISON, C ;

LIEN, EJ ;

ZINGER, AP ;

HUSSAIN, M ;

TONG, GL ;

GOLDEN, M .

JOURNAL OF PHARMACEUTICAL SCIENCES, 1971, 60 (07) :1058-&

[5] MEDIUM RING NITROGEN-HETEROCYCLES [J].

EVANS, PA ;

HOLMES, AB .

TETRAHEDRON, 1991, 47 (44) :9131-9166

[6] A SYNTHESIS OF CYCLIC PEPTIDES UTILIZING HIGH MOLECULAR WEIGHT CARRIERS [J].

FRIDKIN, M ;

PATCHORN.A ;

KATCHALS.E .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1965, 87 (20) :4646-&

[7] NEW USEFUL REAGENTS FOR PEPTIDE-SYNTHESIS - INSOLUBLE ACTIVE ESTERS OF POLYSTYRENE-BOUND 1-HYDROXYBENZOTRIAZOLE [J].

KALIR, R ;

WARSHAWSKY, A ;

FRIDKIN, M ;

PATCHORNIK, A .

EUROPEAN JOURNAL OF BIOCHEMISTRY, 1975, 59 (01) :55-61

[8]

KELLER O, 1984, ORG SYNTH, V63, P160

[9] SEQUENCE DEPENDENCE IN SOLID-PHASE-SYNTHESIS-CYCLIZATION-CLEAVAGE FOR CYCLO(-ARGINYL-GLYCYL-ASPARTYL-PHENYLGLYCYL-) [J].

NISHINO, N ;

XU, M ;

MIHARA, H ;

FUJIMOTO, T ;

UENO, Y ;

KUMAGAI, H .

TETRAHEDRON LETTERS, 1992, 33 (11) :1479-1482

[10] MULTICYCLIC POLYPEPTIDE MODEL COMPOUNDS .1. SYNTHESIS OF A TRICYCLIC AMPHIPHILIC ALPHA-HELICAL PEPTIDE USING AN OXIME RESIN, SEGMENT-CONDENSATION APPROACH [J].

OSAPAY, G ;

TAYLOR, JW .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1990, 112 (16) :6046-6051

← 1 2 →