SYNTHETIC ENKEPHALIN ANALOG WITH PROLONGED PARENTERAL AND ORAL ANALGESIC ACTIVITY

被引:382
作者
ROEMER, D
BUESCHER, HH
HILL, RC
PLESS, J
BAUER, W
CARDINAUX, F
CLOSSE, A
HAUSER, D
HUGUENIN, R
机构
[1] SANDOZ LTD,DIV BIOL & MED RES,CH-4002 BASEL,SWITZERLAND
[2] SANDOZ LTD,DIV CHEM RES PHARMACEUT,CH-4002 BASEL,SWITZERLAND
关键词
D O I
10.1038/268547a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:547 / 549
页数:3
相关论文
共 33 条
  • [1] ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT
    BELLUZZI, JD
    GRANT, N
    GARSKY, V
    SARANTAKIS, D
    WISE, CD
    STEIN, L
    [J]. NATURE, 1976, 260 (5552) : 625 - 626
  • [2] BIRDSALL NJM, 1976, OPIATES ENDOGENOUS O, P19
  • [3] ENDORPHINS - PROFOUND BEHAVIORAL-EFFECTS IN RATS SUGGEST NEW ETIOLOGICAL FACTORS IN MENTAL-ILLNESS
    BLOOM, F
    SEGAL, D
    LING, N
    GUILLEMIN, R
    [J]. SCIENCE, 1976, 194 (4265) : 630 - 632
  • [4] DETERMINING THRESHOLDS OF AVERSIVE BRAIN STIMULATION
    BOREN, JJ
    MALIS, JL
    [J]. AMERICAN JOURNAL OF PHYSIOLOGY, 1961, 201 (03): : 429 - &
  • [5] BRADBURY AF, 1976, OPIATES ENDOGENOUS O, P9
  • [6] EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE
    BUSCHER, HH
    HILL, RC
    ROMER, D
    CARDINAUX, F
    CLOSSE, A
    HAUSER, D
    PLESS, J
    [J]. NATURE, 1976, 261 (5559) : 423 - 425
  • [7] D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
  • [8] SELF-ADMINISTRATION OF PSYCHOACTIVE SUBSTANCES BY MONKEY - A MEASURE OF PSYCHOLOGICAL DEPENDENCE
    DENEAU, G
    YANAGITA, T
    SEEVERS, MH
    [J]. PSYCHOPHARMACOLOGIA, 1969, 16 (01): : 30 - &
  • [9] EDDY NB, 1953, J PHARMACOL EXP THER, V107, P385
  • [10] INDUCTION OF EXCESSIVE GROOMING IN RAT BY FRAGMENTS OF LIPOTROPIN
    GISPEN, WH
    WIEGANT, VM
    BRADBURY, AF
    HULME, EC
    SMYTH, DG
    SNELL, CR
    DEWIED, D
    [J]. NATURE, 1976, 264 (5588) : 794 - 795