SYNTHESIS AND N-SUBSTITUTION OF AN UNCOMMON HETEROCYCLIC SYSTEM - OXAZOLO[5,4-B]PYRIDIN-2(1H)-ONE

被引：14

作者：

FLOUZAT, C ^{[1
]}

BLANCHET, M ^{[1
]}

GUILLAUMET, G ^{[1
]}

机构：

[1] UNIV ORLEANS,CNRS,CHIM BIOORGAN & ANALYT LAB,BP 6759,F-45067 ORLEANS 2,FRANCE

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 32期

关键词：

OXAZOLO[5,4-B]PYRIDIN-2(1H)-ONE; N-SUBSTITUTED OXAZOLO[5,4-B]PYRIDIN-2(1H)-ONES; TRIPHOSGENE;

D O I：

10.1016/S0040-4039(00)61315-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Oxazolo[5,4-b]pyridin-2(1H)-one 2 can be obtained in a one-step procedure. Its reactivity towards nucleophiles and alkylation to nitrogen are described.

引用

页码：4571 / 4574

页数：4

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