CLINICAL-EXPERIENCES WITH TRANDOLAPRIL

被引:12
作者
GAILLARD, CA [1 ]
DELEEUW, PW [1 ]
机构
[1] UNIV LIMBURG HOSP,DEPT MED,POB 5800,6202 AZ MAASTRICHT,NETHERLANDS
关键词
D O I
10.1016/0002-8703(93)90453-G
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
In this article the clinical experiences with the new nonsulphydryl angiotensin-converting enzyme inhibitor trandolapril are reviewed. The drug lowers blood pressure effectively in patients with mild-to-severe hypertension including elderly and obese patients. Distinguishing features of the compound are its long plasma half-life and high degree of lipophilicity.
引用
收藏
页码:1542 / 1546
页数:5
相关论文
共 23 条
[1]  
BACKHOUSE CJ, IN PRESS J CARDIOVAS
[2]  
CESARONE MR, IN PRESS J CARDIOVAS
[3]   DIFFERENTIAL-EFFECTS OF ORAL TRANDOLAPRIL AND ENALAPRIL ON RAT-TISSUE ANGIOTENSIN-CONVERTING ENZYME [J].
CHEVILLARD, C ;
BROWN, NL ;
MATHIEU, MN ;
LALIBERTE, F ;
WORCEL, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 147 (01) :23-28
[4]  
COLLINS JD, 1988, INVESTIGATION PHARMA
[5]   EVIDENCE FOR A SINGLE ACTIVE-SITE IN THE HUMAN ANGIOTENSIN I-CONVERTING ENZYME FROM INHIBITOR BINDING-STUDIES WITH [H-3] RU-44-403 - ROLE OF CHLORIDE [J].
CUMIN, F ;
VELLAUD, V ;
CORVOL, P ;
ALHENCGELAS, F .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1989, 163 (02) :718-725
[6]  
DAVEY A, 1990, UK8957005 REP
[7]  
DEBRUIJN JHB, IN PRESS J CARDIOVAS
[8]  
DELEEUW PW, IN PRESS J CARDIOVAS
[9]   HEMODYNAMIC-EFFECTS OF ANGIOTENSIN-CONVERTING ENZYME-INHIBITORS IN ESSENTIAL-HYPERTENSION - A REVIEW [J].
FITZPATRICK, MA ;
JULIUS, S .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1985, 7 :S35-S39