STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF ACROSIN BY BENZAMIDINE DERIVATIVES

被引：17

作者：

PARRISH, RF

STRAUS, JW

PAULSON, JD

POLAKOSKI, KL

TIDWELL, RR

GERATZ, JD

STEVENS, FM

机构：

[1] WASHINGTON UNIV,SCH MED,DEPT OBSTET & GYNECOL,ST LOUIS,MO 63110

[2] UNIV N CAROLINA,SCH MED,DEPT PATHOL,CHAPEL HILL,NC 27514

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1978年 / 21卷 / 11期

关键词：

D O I：

10.1021/jm00209a008

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1132 / 1136

页数：5

共 25 条

[1] A chemotherapeutic comparison of the trypanocidal action of some aromatic diamidines [J].

Ashley, JN ;

Barber, HJ ;

Ewins, AJ ;

Newbery, G ;

Self, ADH .

JOURNAL OF THE CHEMICAL SOCIETY, 1942, :103-116

[2] THE SEARCH FOR CHEMOTHERAPEUTIC AMIDINES .10. SUBSTITUTED 4-4'-DIAMIDINO-ALPHA-OMEGA-DIPHENOXYALKANES AND 4-4'-DIAMIDINO-ALPHA-OMEGA-DIPHENYL ETHERS [J].

BERG, SS ;

NEWBERY, G .

JOURNAL OF THE CHEMICAL SOCIETY, 1949, (MAR) :642-648

[3]

BHATTACHARYYA AK, 1976, J REPROD FERTIL, V47, P97

[4] DISC ELECTROPHORESIS [J].

BREWER, JM ;

ASHWORTH, RB .

JOURNAL OF CHEMICAL EDUCATION, 1969, 46 (01) :41-&

[5] THE DETERMINATION OF ENZYME INHIBITOR CONSTANTS [J].

DIXON, M .

BIOCHEMICAL JOURNAL, 1953, 55 (01) :170-171

[6] IMPROVED ZYMOGRAPHIC DETECTION OF BOVINE ACROSIN [J].

GARNER, DL .

ANALYTICAL BIOCHEMISTRY, 1975, 67 (02) :688-694

[7] NOVEL BIS(BENZAMIDINO) COMPOUNDS WITH AN AROMATIC CENTRAL LINK - INHIBITORS OF THROMBIN, PANCREATIC KALLIKREIN, TRYPSIN, AND COMPLEMENT [J].

GERATZ, JD ;

CHENG, MCF ;

TIDWELL, RR .

JOURNAL OF MEDICINAL CHEMISTRY, 1976, 19 (05) :634-639

[8] NEW AROMATIC DIAMIDINES WITH CENTRAL ALPHA-OXYALKANE OR ALPHA,OMEGA-DIOXYALKANE CHAINS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TRYPSIN, PANCREATIC KALLIKREIN, AND THROMBIN AND FOR INHIBITION OF OVERALL COAGULATION PROCESS [J].

GERATZ, JD ;

CHENG, MCF ;

TIDWELL, RR .

JOURNAL OF MEDICINAL CHEMISTRY, 1975, 18 (05) :477-481

[9] DIAMIDINO-ALPHA, OMEGO-DIPHENOXYALKANES - STRUCTURE-ACTIVITY RELATIONSHIPS FOR INHIBITION OF THROMBIN, PANCREATIC KALLIKREIN, AND TRYPSIN [J].

GERATZ, JD ;

WHITMORE, AC ;

CHENG, MCF ;

PIANTADOSI, C .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (09) :970-975

[10]

GERATZ JD, 1977, CHEM BIOL THROMBIN, P179

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