INHIBITION OF PERIPHERAL AROMATIZATION BY AROMATASE INHIBITORS, 4-HYDROXY-ANDROSTENE-3,17-DIONE AND 4-ACETOXY-ANDROSTENE-3,17-DIONE

被引:95
作者
BRODIE, AMH [1 ]
LONGCOPE, C [1 ]
机构
[1] WORCESTER FDN EXPTL BIOL,SHREWSBURY,MA 01545
关键词
D O I
10.1210/endo-106-1-19
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:19 / 21
页数:3
相关论文
共 14 条
[1]  
BAIRD D, 1968, PERSPECT BIOL MED, V11, P384
[2]   AROMATASE INHIBITORS .4. REGRESSION OF HORMONE-DEPENDENT, MAMMARY-TUMORS IN THE RAT WITH 4-ACETOXY-4-ANDROSTENE-3,17-DIONE [J].
BRODIE, AMH ;
MARSH, D ;
BRODIE, HJ .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1979, 10 (04) :423-429
[3]   AROMATASE INHIBITORS .3. STUDIES ON ANTI-FERTILITY EFFECT OF 4-ACETOXY-4-ANDROSTENE-3,17-DIONE [J].
BRODIE, AMH ;
WU, JT ;
MARSH, DA ;
BRODIE, HJ .
BIOLOGY OF REPRODUCTION, 1978, 18 (03) :365-370
[4]   EFFECT OF AN AROMATASE INHIBITOR, 4-HYDROXY-4-ANDROSTENE-3,17-DIONE, ON ESTROGEN-DEPENDENT PROCESSES IN REPRODUCTION AND BREAST-CANCER [J].
BRODIE, AMH ;
SCHWARZEL, WC ;
SHAIKH, AA ;
BRODIE, HJ .
ENDOCRINOLOGY, 1977, 100 (06) :1684-1695
[5]   PLASMA PRECURSORS OF ESTROGEN .2. CORRELATION OF EXTENT OF CONVERSION OF PLASMA ANDROSTENEDIONE TO ESTRONE WITH AGE [J].
HEMSELL, DL ;
GRODIN, JM ;
BRENNER, PF ;
SIITERI, PK ;
MACDONALD, PC .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1974, 38 (03) :476-479
[6]   STEROID METABOLISM BY HUMAN MAMMARY-CARCINOMA [J].
LI, K ;
CHANDRA, DP ;
FOO, T ;
ADAMS, JB ;
MCDONALD, D .
STEROIDS, 1976, 28 (04) :561-574
[7]   AROMATIZATION OF ANDROGENS BY MUSCLE AND ADIPOSE-TISSUE INVIVO [J].
LONGCOPE, C ;
PRATT, JH ;
SCHNEIDER, SH ;
FINEBERG, SE .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1978, 46 (01) :146-152
[9]   PLASMA PRECURSORS OF ESTROGEN .I. EXTENT OF CONVERSION OF PLASMA DELTA4-ANDROSTENEDIONE TO ESTRONE IN NORMAL MALES AND NONPREGNANT NORMAL CASTRATE AND ADRENALECTOMIZED FEMALES [J].
MACDONALD, PC ;
ROMBAUT, RP ;
SIITERI, PK .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1967, 27 (08) :1103-+
[10]  
MILLER WR, 1974, LANCET, V2, P866