SYNTHESES OF BENZOMORPHAN AND RELATED COMPOUNDS .I. SYNTHESIS OF N-SUBSTITUTED-1,2,3,4,5,6-HEXAHYDRO-8-HYDROXY-2,6-METHANO-6,11-DIMETHYL-3 BENZAZOCINE [STUDIES ON SYNTHESES OF HETEROCYCLIC COMPOUNDS .282.]

被引：36

作者：

KAMETANI, T

KIGASAWA, K

HIIRAGI, M

HAYASAKA, T

WAGATSUM.N

WAKISAKA, K

机构：

[1] Pharmaceutical Institute, School of Medicine, Tohoku University and Research Laboratories, Grelan Pharamaceutical Co, Ltd., Sendai

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1969年 / 6卷 / 01期

关键词：

D O I：

10.1002/jhet.5570060108

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A modified synthesis of pentazocine, l,2,3,4,5,6‐hexahydro‐8‐hydroxy‐2,6‐methano‐6, H‐dimethyl‐3‐(3‐methyl‐2‐butenyl)‐3‐benzazocine (III), has been achieved and catalytic hydro‐genation has been found to be effective for the debenzylation of quaternary ammonium salts. Copyright © 1969 Journal of Heterocyclic Chemistry

引用

页码：43 / &

共 17 条

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[9] STRUCTURES RELATED TO MORPHINE .11. ANALOGS AND A DIASTEREOISOMER OF 2'-HYDROXY-2,5,9-TRIMETHYL-6,7-BENZOMORPHAN
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