BQ-123, A SELECTIVE ENDOTHELIN ET(A) RECEPTOR ANTAGONIST

被引:27
作者
MORELAND, S [1 ]
机构
[1] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT PHARMACOL,PRINCETON,NJ 08543
来源
CARDIOVASCULAR DRUG REVIEWS | 1994年 / 12卷 / 01期
关键词
BQ-123; ENDOTHELIN; ENDOTHELIN RECEPTOR ANTAGONIST;
D O I
10.1111/j.1527-3466.1994.tb00283.x
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:48 / 69
页数:22
相关论文
共 196 条
[21]  
CAI H, 1992, CLIN RES, V40, pA807
[22]   EFFECT OF AN ENDOTHELIN-RECEPTOR ANTAGONIST ON ISCHEMIC ACUTE-RENAL-FAILURE [J].
CHAN, L ;
CHITTINANDANA, A ;
SHAPIRO, JI ;
SHANLEY, PF ;
SCHRIER, RW .
AMERICAN JOURNAL OF PHYSIOLOGY, 1994, 266 (01) :F135-F138
[23]   ENDOTHELIN INHIBITS BASAL AND STIMULATED RELEASE OF PROLACTIN BY HUMAN DECIDUAL CELLS [J].
CHAO, HS ;
MYERS, SE ;
HANDWERGER, S .
ENDOCRINOLOGY, 1993, 133 (02) :505-510
[24]  
CHEN SJ, 1993, FASEB J, V7, pA649
[25]   SHORT-TERM REGULATION OF ENDOTHELIN RECEPTOR-MEDIATED PHOSPHOINOSITIDE HYDROLYSIS AND ARACHIDONIC-ACID RELEASE IN A7R5 SMOOTH-MUSCLE CELLS [J].
CIOFFI, CL ;
GARAY, M .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 22 :S168-S170
[26]  
CIOFFI CL, 1992, J PHARMACOL EXP THER, V262, P611
[27]   BQ-123, A PEPTIDIC ENDOTHELIN ETA RECEPTOR ANTAGONIST, PREVENTS THE EARLY CEREBRAL VASOSPASM FOLLOWING SUBARACHNOID HEMORRHAGE AFTER INTRACISTERNAL BUT NOT INTRAVENOUS-INJECTION [J].
CLOZEL, M ;
WATANABE, H .
LIFE SCIENCES, 1993, 52 (09) :825-834
[28]   EVIDENCE FOR AN EFFECTOR ROLE OF ENDOTHELIN IN CLOSURE OF THE DUCTUS-ARTERIOSUS AT BIRTH [J].
COCEANI, F ;
KELSEY, L ;
SEIDLITZ, E .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1992, 70 (07) :1061-1064
[29]   A CONFORMATIONAL STUDY BY H-1-NMR OF A CYCLIC PENTAPEPTIDE ANTAGONIST OF ENDOTHELIN [J].
COLES, M ;
SOWEMIMO, V ;
SCANLON, D ;
MUNRO, SLA ;
CRAIK, DJ .
JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (18) :2658-2665
[30]   IMPLICATION OF DIFFERENT ENDOTHELIN RECEPTORS IN THE VASCULAR ACTION OF A HYPERTENSIVE DOSE OF ET-1 IN RAT [J].
CORNET, S ;
PIROTZKY, E ;
BRAQUET, P .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 22 :S239-S292