DILTIAZEM PHARMACOKINETICS IN THE RAT AND RELATIONSHIP BETWEEN ITS SERUM CONCENTRATION AND UTERINE AND CARDIOVASCULAR EFFECTS

被引:14
作者
DOWNING, SJ [1 ]
EDWARDS, D [1 ]
HOLLINGSWORTH, M [1 ]
机构
[1] UNIV MANCHESTER,DEPT PHYSIOL SCI,SMOOTH MUSCLE RES GRP,OXFORD RD,MANCHESTER M13 9PT,LANCS,ENGLAND
关键词
D O I
10.1111/j.1476-5381.1987.tb11271.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:735 / 745
页数:11
相关论文
共 21 条
[1]   THE POTENCIES AND SELECTIVITIES OF 4 CALCIUM-ANTAGONISTS AS INHIBITORS OF UTERINE CONTRACTIONS IN THE RAT INVIVO [J].
ABEL, MH ;
HOLLINGSWORTH, M .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 85 (01) :263-269
[2]   THE EFFECTS OF LONG-TERM INFUSION OF SALBUTAMOL, DILTIAZEM AND NIFEDIPINE ON UTERINE CONTRACTIONS IN THE OVARIECTOMIZED, POSTPARTUM RAT [J].
ABEL, MH ;
HOLLINGSWORTH, M .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 88 (03) :577-584
[3]  
ABEL MH, 1986, J REPROD FERTIL, V77, P559
[4]   CHANGES IN WATER AND ELECTROLYTE BALANCE, PLASMA-VOLUME AND COMPOSITION DURING PREGNANCY IN THE RAT [J].
ATHERTON, JC ;
DARK, JM ;
GARLAND, HO ;
MORGAN, MRA ;
PIDGEON, J ;
SONI, S .
JOURNAL OF PHYSIOLOGY-LONDON, 1982, 330 (SEP) :81-93
[5]   MECHANISMS OF ACTION OF TRANSMITTERS AND OTHER SUBSTANCES ON SMOOTH-MUSCLE [J].
BOLTON, TB .
PHYSIOLOGICAL REVIEWS, 1979, 59 (03) :606-718
[6]  
BOX MJ, 1969, MONOGRAPH IMPERIAL C, V5
[7]  
DOWNING S J, 1986, British Journal of Pharmacology, V89, p620P
[8]   NEED FOR CALCIUM IN CONTRACTILE RESPONSES INDUCED BY ACETYLCHOLINE AND POTASSIUM IN RAT UTERUS [J].
EDMAN, KAP ;
SCHILD, HO .
JOURNAL OF PHYSIOLOGY-LONDON, 1962, 161 (03) :424-&
[9]   THE SPASMOGENIC ACTION OF OXYTOCIN IN THE RAT UTERUS COMPARISON WITH OTHER AGONISTS [J].
EDWARDS, D ;
GOOD, DM ;
GRANGER, SE ;
HOLLINGSWORTH, M ;
ROBSON, A ;
SMALL, RC ;
WESTON, AH .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 88 (04) :899-908
[10]   EFFECTS OF CALCIUM ENTRY BLOCKERS ON TENSION DEVELOPMENT AND CALCIUM INFLUX IN RAT UTERUS [J].
GRANGER, SE ;
HOLLINGSWORTH, M ;
WESTON, AH .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 87 (01) :147-156