A NEW ROUTE TO 2-ARYL-4-QUINOLONES VIA PALLADIUM CATALYZED CARBONYLATIVE COUPLING OF ORTHO-IODOANILINES WITH TERMINAL ARYLACETYLENES

被引：83

作者：

KALININ, VN

SHOSTAKOVSKY, MV

PONOMARYOV, AB

机构：

[1] Nesmeyanov Institute of Organoelement Compounds, 117813 Moscow

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 03期

关键词：

D O I：

10.1016/S0040-4039(00)74135-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

O-Iodoanilines undergo Pd-catalyzed intramolecular heterocyclization with terminal arylacetylenes in the presence of carbon monoxide to give 2-aryl-4-quinolones.

引用

页码：373 / 376

页数：4

共 12 条

[1]

BARDAMOVA MI, 1982, IZ AKAD NAUK SSSR K, P1184

[2]

BUMAGIN NA, 1984, SYNTHESIS-STUTTGART, P728

[3]

CHEN BC, 1987, SYNTHESIS-STUTTGART, P482

[4]

HIRAKI U, Patent No. 287951

[5]

KASAHARA A, 1981, CHEM IND-LONDON, P121

[6] GENERAL SYNTHESIS OF TERMINAL AND INTERNAL ARYLALKYNES BY PALLADIUM-CATALYZED REACTION OF ALKYNYLZINC REAGENTS WITH ARYL HALIDES [J].

KING, AO ;

NEGISHI, EI ;

VILLANI, FJ ;

SILVEIRA, A .

JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (02) :358-360

[7] SYNTHESIS OF 4-HYDROXYQUINOLINES .6. SYNTHESIS OF 3-NORMAL-HEPTYL-7-METHOXY-2-METHYL-4-QUINOLINOL [J].

LEONARD, NJ ;

HERBRANDSON, HF ;

VANHEYNINGEN, EM .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1946, 68 (07) :1279-1281

[8]

OSAWA T, Patent No. 343547

[9] THE CHEMISTRY OF 4-HYDROXYQUINOLINES [J].

REITSEMA, RH .

CHEMICAL REVIEWS, 1948, 43 (01) :43-68

[10] REACTION BETWEEN BETA-KETO ESTERS AND ARYLAMINES IN PRESENCE OF POLYPHOSPHORIC ACID .1. ETHYL BENZOYLACETATE AND ARYLAMINES [J].

STASKUN, B ;

ISRAELSTAM, SS .

JOURNAL OF ORGANIC CHEMISTRY, 1961, 26 (09) :3191-&

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