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THE PHYSICOCHEMICAL APPROACH TO DRUG DESIGN AND DISCOVERY (QSAR)
被引:58
作者
:
HANSCH, C
论文数:
0
引用数:
0
h-index:
0
HANSCH, C
机构
:
来源
:
DRUG DEVELOPMENT RESEARCH
|
1981年
/ 1卷
/ 04期
关键词
:
D O I
:
10.1002/ddr.430010403
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:267 / 309
页数:43
相关论文
共 134 条
[1]
ARIENS EJ, 1971, DRUG DESIGN, V1, P133
[2]
FURTHER EVALUATION OF A QUANTITATIVE MATHEMATICAL-MODEL FOR PREDICTING ACUTE TOXICITY OF ACRYLATE AND METHACRYLATE ESTERS
BASS, GE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
BASS, GE
LAWRENCE, WH
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
LAWRENCE, WH
PURCELL, WP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
PURCELL, WP
AUTIAN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
AUTIAN, J
[J].
JOURNAL OF DENTAL RESEARCH,
1974,
53
(03)
: 756
-
756
[3]
AN EXAMPLE OF SUCCESSFUL PREDICTION OF CHOLINESTERASE INHIBITORY POTENCY FROM REGRESSION ANALYSIS
BEASLEY, JG
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Medicinal Chemistry, College of Pharmacy, University of Tennessee Medical Units, Memphis
BEASLEY, JG
PURCELL, WP
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Medicinal Chemistry, College of Pharmacy, University of Tennessee Medical Units, Memphis
PURCELL, WP
[J].
BIOCHIMICA ET BIOPHYSICA ACTA,
1969,
178
(01)
: 175
-
&
[4]
COMPOUNDS DESIGNED TO FIT A SITE OF KNOWN STRUCTURE IN HUMAN HEMOGLOBIN
BEDDELL, CR
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
BEDDELL, CR
GOODFORD, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
GOODFORD, PJ
NORRINGTON, FE
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
NORRINGTON, FE
WILKINSON, S
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WILKINSON, S
WOOTTON, R
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WOOTTON, R
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1976,
57
(02)
: 201
-
209
[5]
Studies in chemotherapy. VII. A theory of the relation of structure to activity of sulfanilamide type compounds
Bell, PH
论文数:
0
引用数:
0
h-index:
0
机构:
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
Bell, PH
Roblin, RO
论文数:
0
引用数:
0
h-index:
0
机构:
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
Roblin, RO
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1942,
64
: 2905
-
2917
[6]
CORRELATION OF SERUM BINDING OF PENICILLINS WITH PARTITION COEFFICIENTS
BIRD, AE
论文数:
0
引用数:
0
h-index:
0
BIRD, AE
MARSHALL, AC
论文数:
0
引用数:
0
h-index:
0
MARSHALL, AC
[J].
BIOCHEMICAL PHARMACOLOGY,
1967,
16
(12)
: 2275
-
&
[7]
ANTIALLERGIC ACTIVITY OF 2-PHENYL-8-AZAPURIN-6-ONES
BROUGHTON, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
BROUGHTON, BJ
CHAPLEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
CHAPLEN, P
KNOWLES, P
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
KNOWLES, P
LUNT, E
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
LUNT, E
MARSHALL, SM
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MARSHALL, SM
PAIN, DL
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
PAIN, DL
WOOLDRIDGE, KRH
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
WOOLDRIDGE, KRH
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1975,
18
(11)
: 1117
-
1122
[8]
A CORRELATION OF THYROXINE-LIKE ACTIVITY AND CHEMICAL STRUCTURE
BRUICE, TC
论文数:
0
引用数:
0
h-index:
0
BRUICE, TC
KHARASCH, N
论文数:
0
引用数:
0
h-index:
0
KHARASCH, N
WINZLER, RJ
论文数:
0
引用数:
0
h-index:
0
WINZLER, RJ
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1956,
62
(02)
: 305
-
317
[9]
BUCHI J, 1975, ARZNEIM FORSCH, V25, P1233
[10]
PREDICTABILITY OF CORRELATIONS BETWEEN IN-VITRO TETRACYCLINE POTENCIES AND SUBSTITUENT INDICES
CAMMARAT.A
论文数:
0
引用数:
0
h-index:
0
CAMMARAT.A
YAU, SJ
论文数:
0
引用数:
0
h-index:
0
YAU, SJ
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1970,
13
(01)
: 93
-
&
←
1
2
3
4
5
6
7
8
9
10
→
共 134 条
[1]
ARIENS EJ, 1971, DRUG DESIGN, V1, P133
[2]
FURTHER EVALUATION OF A QUANTITATIVE MATHEMATICAL-MODEL FOR PREDICTING ACUTE TOXICITY OF ACRYLATE AND METHACRYLATE ESTERS
BASS, GE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
BASS, GE
LAWRENCE, WH
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
LAWRENCE, WH
PURCELL, WP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
PURCELL, WP
AUTIAN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TENNESSEE,MED UNITS,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MEMPHIS,TN 38163
AUTIAN, J
[J].
JOURNAL OF DENTAL RESEARCH,
1974,
53
(03)
: 756
-
756
[3]
AN EXAMPLE OF SUCCESSFUL PREDICTION OF CHOLINESTERASE INHIBITORY POTENCY FROM REGRESSION ANALYSIS
BEASLEY, JG
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Medicinal Chemistry, College of Pharmacy, University of Tennessee Medical Units, Memphis
BEASLEY, JG
PURCELL, WP
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Medicinal Chemistry, College of Pharmacy, University of Tennessee Medical Units, Memphis
PURCELL, WP
[J].
BIOCHIMICA ET BIOPHYSICA ACTA,
1969,
178
(01)
: 175
-
&
[4]
COMPOUNDS DESIGNED TO FIT A SITE OF KNOWN STRUCTURE IN HUMAN HEMOGLOBIN
BEDDELL, CR
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
BEDDELL, CR
GOODFORD, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
GOODFORD, PJ
NORRINGTON, FE
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
NORRINGTON, FE
WILKINSON, S
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WILKINSON, S
WOOTTON, R
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WELLCOME RES LABS,BECKENHAM,KENT,ENGLAND
WOOTTON, R
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1976,
57
(02)
: 201
-
209
[5]
Studies in chemotherapy. VII. A theory of the relation of structure to activity of sulfanilamide type compounds
Bell, PH
论文数:
0
引用数:
0
h-index:
0
机构:
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
Bell, PH
Roblin, RO
论文数:
0
引用数:
0
h-index:
0
机构:
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
American Cyanamid Co, Stamford Res Labs, Stamford, CT USA
Roblin, RO
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1942,
64
: 2905
-
2917
[6]
CORRELATION OF SERUM BINDING OF PENICILLINS WITH PARTITION COEFFICIENTS
BIRD, AE
论文数:
0
引用数:
0
h-index:
0
BIRD, AE
MARSHALL, AC
论文数:
0
引用数:
0
h-index:
0
MARSHALL, AC
[J].
BIOCHEMICAL PHARMACOLOGY,
1967,
16
(12)
: 2275
-
&
[7]
ANTIALLERGIC ACTIVITY OF 2-PHENYL-8-AZAPURIN-6-ONES
BROUGHTON, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
BROUGHTON, BJ
CHAPLEN, P
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
CHAPLEN, P
KNOWLES, P
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
KNOWLES, P
LUNT, E
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
LUNT, E
MARSHALL, SM
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MARSHALL, SM
PAIN, DL
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
PAIN, DL
WOOLDRIDGE, KRH
论文数:
0
引用数:
0
h-index:
0
机构:
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
MAY & BAKER LTD,RES LABS,DAGENHAM,ESSEX,ENGLAND
WOOLDRIDGE, KRH
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1975,
18
(11)
: 1117
-
1122
[8]
A CORRELATION OF THYROXINE-LIKE ACTIVITY AND CHEMICAL STRUCTURE
BRUICE, TC
论文数:
0
引用数:
0
h-index:
0
BRUICE, TC
KHARASCH, N
论文数:
0
引用数:
0
h-index:
0
KHARASCH, N
WINZLER, RJ
论文数:
0
引用数:
0
h-index:
0
WINZLER, RJ
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1956,
62
(02)
: 305
-
317
[9]
BUCHI J, 1975, ARZNEIM FORSCH, V25, P1233
[10]
PREDICTABILITY OF CORRELATIONS BETWEEN IN-VITRO TETRACYCLINE POTENCIES AND SUBSTITUENT INDICES
CAMMARAT.A
论文数:
0
引用数:
0
h-index:
0
CAMMARAT.A
YAU, SJ
论文数:
0
引用数:
0
h-index:
0
YAU, SJ
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1970,
13
(01)
: 93
-
&
←
1
2
3
4
5
6
7
8
9
10
→