THE NUCLEAR UPTAKE OF 6-ALPHA-[H-3]METHYLPROGESTERONE AND ITS 20-ALPHA-HYDROXY METABOLITE - THE REQUIREMENT FOR MULTIPLE RECEPTORS

被引:7
作者
BROWN, TR [1 ]
BULLOCK, LP [1 ]
BARDIN, CW [1 ]
机构
[1] PENN STATE UNIV,MILTON S HERSHEY MED CTR,DEPT CHEM,DIV ENDOCRINOL,HERSHEY,PA 17033
关键词
D O I
10.1210/endo-109-6-1821
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:1821 / 1829
页数:9
相关论文
共 30 条
[1]   HUMAN LIVER NUCLEAR TRANSCORTIN - ITS POSTULATED ROLE IN GLUCOCORTICOID REGULATION OF GENETIC ACTIVITY [J].
AMARAL, L ;
LIN, K ;
SAMUELS, AJ ;
WERTHAMER, S .
BIOCHIMICA ET BIOPHYSICA ACTA, 1974, 362 (02) :332-345
[2]  
Bardin C W, 1973, Recent Prog Horm Res, V29, P65
[3]   TESTOSTERONE - A MAJOR DETERMINANT OF EXTRA-GENITAL SEXUAL DIMORPHISM [J].
BARDIN, CW ;
CATTERALL, JF .
SCIENCE, 1981, 211 (4488) :1285-1294
[4]   INTERACTION OF GLUCOCORTICOIDS WITH RAT-LIVER NUCLEI - EFFECT OF ADRENALECTOMY AND CORTISOL ADMINISTRATION [J].
BEATO, M ;
KALIMI, M ;
BEATO, W ;
FEIGELSO.P .
ENDOCRINOLOGY, 1974, 94 (02) :377-387
[5]   THE BIOLOGICAL ACTIONS AND METABOLISM OF 6-ALPHA-METHYLPROGESTERONE - A PROGESTIN THAT MIMICS AND MODIFIES THE EFFECTS OF TESTOSTERONE [J].
BROWN, TR ;
BULLOCK, LP ;
BARDIN, CW .
ENDOCRINOLOGY, 1981, 109 (06) :1814-1820
[6]   INVITRO AND INVIVO BINDING OF PROGESTINS TO THE ANDROGEN RECEPTOR OF MOUSE KIDNEY - CORRELATION WITH BIOLOGICAL-ACTIVITIES [J].
BROWN, TR ;
BULLOCK, L ;
BARDIN, CW .
ENDOCRINOLOGY, 1979, 105 (06) :1281-1287
[7]   EFFECT OF PROGESTINS ON SUBMAXILLARY-GLAND EPIDERMAL GROWTH-FACTOR - DEMONSTRATION OF ANDROGENIC, SYNANDROGENIC AND ANTIANDROGENIC ACTIONS [J].
BULLOCK, LP ;
BARTHE, PL ;
MOWSZOWICZ, I ;
ORTH, DN ;
BARDIN, CW .
ENDOCRINOLOGY, 1975, 97 (01) :189-195
[8]   INVIVO ANDROGEN RETENTION IN MOUSE KIDNEY [J].
BULLOCK, LP ;
BARDIN, CW .
STEROIDS, 1975, 25 (01) :107-119
[9]   ANDROGENIC, ANTI-ANDROGENIC, AND SYNANDROGENIC ACTIONS OF PROGESTINS - ROLE OF STERIC AND ALLOSTERIC INTERACTIONS WITH ANDROGEN RECEPTORS [J].
BULLOCK, LP ;
BARDIN, CW ;
SHERMAN, MR .
ENDOCRINOLOGY, 1978, 103 (05) :1768-1782
[10]  
BULLOCK LP, 1977, PHARM STEROID CONTRA, P353