THE DISCOVERY OF SULFONAMIDE ENDOTHELIN ANTAGONISTS AND THE DEVELOPMENT OF THE ORALLY-ACTIVE ET(A) ANTAGONIST 5-(DIMETHYLAMINO)-N-(3,4-DIMETHYL-5-ISOXAZOLYL)-1-NAPHTHALENESULFONAMIDE

被引：141

作者：

STEIN, PD

HUNT, JT

FLOYD, DM

MORELAND, S

DICKINSON, KEJ

MITCHELL, C

LIU, ECK

WEBB, ML

MURUGESAN, N

DICKEY, J

MCMULLEN, D

ZHANG, RG

LEE, VG

SERAFINO, R

DELANEY, C

SCHAEFFER, TR

KOZLOWSKI, M

机构：

[1] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT CHEM CARDIOVASC AGENTS,PRINCETON,NJ 08543

[2] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT CARDIOVASC BIOCHEM,PRINCETON,NJ 08543

[3] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT PHARMACOL,PRINCETON,NJ 08543

[4] BRISTOL MYERS SQUIBB CO,PHARMACEUT RES INST,DEPT BIOMOLEC SCREENING,WALLINGFORD,CT 06492

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 03期

关键词：

D O I：

10.1021/jm00029a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：329 / 331

页数：3

共 29 条

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