CHARACTERIZATION OF [H-3] QUIPAZINE BINDING TO 5-HYDROXYTRYPTAMINE3 RECEPTORS IN RAT-BRAIN MEMBRANES

被引:67
作者
MILBURN, CM [1 ]
PEROUTKA, SJ [1 ]
机构
[1] STANFORD UNIV,MED CTR,DEPT NEUROL,C-338,STANFORD,CA 94305
关键词
D O I
10.1111/j.1471-4159.1989.tb07258.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1787 / 1792
页数:6
相关论文
共 27 条
[1]   PROPOSALS FOR THE CLASSIFICATION AND NOMENCLATURE OF FUNCTIONAL RECEPTORS FOR 5-HYDROXYTRYPTAMINE [J].
BRADLEY, PB ;
ENGEL, G ;
FENIUK, W ;
FOZARD, JR ;
HUMPHREY, PPA ;
MIDDLEMISS, DN ;
MYLECHARANE, EJ ;
RICHARDSON, BP ;
SAXENA, PR .
NEUROPHARMACOLOGY, 1986, 25 (06) :563-576
[2]   5-HYDROXYTRYPTAMINE RECEPTORS IN MOUSE DUODENUM [J].
DRAKONTIDES, AB ;
GERSHON, MD .
BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (03) :480-+
[3]  
FAKE C S, 1987, British Journal of Pharmacology, V91, p335P
[4]   PHARMACOLOGICAL PROPERTIES OF PHENYLDIGUANIDE AND OTHER AMIDINE DERIVATIVES IN RELATION TO THOSE OF 5-HYDROXYTRYPTAMINE [J].
FASTIER, FN ;
MCDOWALL, MA ;
WAAL, H .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (04) :527-535
[5]   INDAZOLES AS INDOLE BIOISOSTERES - SYNTHESIS AND EVALUATION OF THE TROPANYL ESTER AND AMIDE OF INDAZOLE-3-CARBOXYLATE AS ANTAGONISTS AT THE SEROTONIN 5HT3 RECEPTOR [J].
FLUDZINSKI, P ;
EVRARD, DA ;
BLOOMQUIST, WE ;
LACEFIELD, WB ;
PFEIFER, W ;
JONES, ND ;
DEETER, JB ;
COHEN, ML .
JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (09) :1535-1537
[6]   5-HT - THE ENIGMA VARIATIONS [J].
FOZARD, JR .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1987, 8 (12) :501-506
[8]  
FOZARD JR, 1977, BRIT J PHARMACOL, V61, pP130
[9]   DIFFERENTIATION OF PRESYNAPTIC AND POSTSYNAPTIC HIGH-AFFINITY SEROTONIN RECEPTOR-BINDING SITES USING PHYSICOCHEMICAL PARAMETERS AND MODIFYING AGENTS [J].
HALL, MD ;
GOZLAN, H ;
EMERIT, MB ;
ELMESTIKAWY, S ;
PICHAT, L ;
HAMON, M .
NEUROCHEMICAL RESEARCH, 1986, 11 (06) :891-912
[10]   IDENTIFICATION OF SEROTONIN 5-HT3 RECOGNITION SITES BY RADIOLIGAND BINDING IN NG108-15 NEUROBLASTOMA-GLIOMA CELLS [J].
HOYER, D ;
NEIJT, HC .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 143 (02) :291-292