ON THE REACTION BETWEEN 3H-1,2-DITHIOLO[3,4-B]-PYRIDINE-3-THIONE AND PRIMARY ALKYL AND ARYLALKLAMINES

被引：25

作者：

BORGNA, P ^{[1
]}

PREGNOLATO, M ^{[1
]}

INVERNIZZI, AG ^{[1
]}

MELLERIO, G ^{[1
]}

机构：

[1] UNIV PAVIA,DIPARTIMENTO CHIM ORGAN,I-27100 PAVIA,ITALY

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1993年 / 30卷 / 04期

关键词：

D O I：

10.1002/jhet.5570300441

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

3H-1,2-Dithiolo[3,4-b]pyridine-3-thione (10) reacts with primary alkylamines to give 1,2-dihydro-2-thioxo-3-pyridinecarbothioamides 11a-g and two minor products. Isothiazolo[5,4-b]pyridine-3(2H)-thiones 12a-g and 3-imino-3H-1,2-dithiolo[3,4-b]pyridines 13a-g were isolated and characterized. Further investigations allowed the synthesis of 12 and 13 in good yield.

引用

页码：1079 / 1084

页数：6

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