C3-METHYLATED 5-HYDROXY-2-(DIPROPYLAMINO)TETRALINS - CONFORMATIONAL AND STERIC PARAMETERS OF IMPORTANCE FOR CENTRAL DOPAMINE RECEPTOR ACTIVATION

被引：20

作者：

JOHANSSON, AM

NILSSON, JLG

KARLEN, A

HACKSELL, U

SVENSSON, K

CARLSSON, A

KENNE, L

SUNDELL, S

机构：

[1] GOTHENBURG UNIV,DEPT PHARMACOL,S-40033 GOTHENBURG,SWEDEN

[2] GOTHENBURG UNIV,DEPT STRUCT CHEM,S-40033 GOTHENBURG,SWEDEN

[3] KABIVITRUM,DEPT ANALYT CHEM,S-11287 STOCKHOLM,SWEDEN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 07期

关键词：

D O I：

10.1021/jm00390a004

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1135 / 1144

页数：10

共 53 条

[1]

Allinger N. L., 1980, QCPE, P395

[2] ADRENERGIC MECHANISMS [J].

ANDEN, NE ;

CARLSSON, A ;

HAGGENDAL, J .

ANNUAL REVIEW OF PHARMACOLOGY, 1969, 9 :119-+

[3]

BEURSKENS PT, 1981, 19812 CRYST LAB TECH

[4]

Cannon J G, 1985, Prog Drug Res, V29, P303

[5] AGONIST-ANTAGONIST INTERACTION ON DOPAMINE RECEPTORS IN BRAIN, AS REFLECTED IN RATES OF TYROSINE AND TRYPTOPHAN HYDROXYLATION [J].

CARLSSON, A ;

KEHR, W ;

LINDQVIST, M .

JOURNAL OF NEURAL TRANSMISSION, 1977, 40 (02) :99-113

[6]

CARLSSON A, 1978, PSYCHOPHARMACOLOGY G, P1057

[7]

Colpaert F C, 1976, Int Rev Neurobiol, V19, P225, DOI 10.1016/S0074-7742(08)60705-9

[8] RELATIVISTIC CALCULATION OF ANOMALOUS SCATTERING FACTORS FOR X-RAYS [J].

CROMER, DT ;

LIBERMAN, D .

JOURNAL OF CHEMICAL PHYSICS, 1970, 53 (05) :1891-&

[9] X-RAY SCATTERING FACTORS COMPUTED FROM NUMERICAL HARTREE-FOCK WAVE FUNCTIONS [J].

CROMER, DT ;

MANN, JB .

ACTA CRYSTALLOGRAPHICA SECTION A-CRYSTAL PHYSICS DIFFRACTION THEORETICAL AND GENERAL CRYSTALLOGRAPHY, 1968, A 24 :321-&

[10] CONFORMATIONAL REQUIREMENTS FOR NOREPINEPHRINE UPTAKE INHIBITION BY PHENETHYLAMINES IN BRAIN SYNAPTOSOMES - EFFECTS OF ALPHA-ALKYL SUBSTITUTION [J].

DEJONG, AP ;

FESIK, SW ;

MAKRIYANNIS, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) :1438-1441

← 1 2 3 4 5 6 →