THE EFFECT OF TEMPERATURE AND CHLORIDE-IONS ON THE STIMULATION OF [FLUNITRAZEPAM-H-3 BINDING BY THE MUSCIMOL ANALOGS THIP AND PIPERIDINE-4-SULFONIC ACID

被引:44
作者
SUPAVILAI, P [1 ]
KAROBATH, M [1 ]
机构
[1] VIENNA UNIV,PSYCHIAT KLIN,DEPT BIOCHEM PSYCHIAT,A-1090 VIENNA,AUSTRIA
关键词
D O I
10.1016/0304-3940(80)90284-0
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:337 / 341
页数:5
相关论文
共 15 条
[1]   MUSCIMOL AND RELATED GABA RECEPTOR AGONISTS - POTENCY OF GABAERGIC DRUGS INVIVO DETERMINED AFTER INTRANIGRAL INJECTION [J].
ARNT, J ;
SCHEELKRUGER, J ;
MAGELUND, G ;
KROGSGAARDLARSEN, P .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1979, 31 (05) :306-313
[2]   PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M ;
KROGSGAARDLARSEN, P ;
FALCH, E .
NATURE, 1979, 280 (5720) :331-333
[3]  
BRILEY MS, 1978, EUR J PHARMACOL, V52, P124
[4]   MODULATION OF BENZODIAZEPINE BINDING-SITES IN CALF CORTEX BY AN ENDOGENOUS FACTOR AND GABAERGIC LIGANDS [J].
DUDAI, Y .
BRAIN RESEARCH, 1979, 167 (02) :422-425
[5]   IS STIMULATION OF BENZODIAZEPINE RECEPTOR-BINDING MEDIATED BY A NOVEL GABA RECEPTOR [J].
KAROBATH, M ;
PLACHETA, P ;
LIPPITSCH, M ;
LARSEN, PK .
NATURE, 1979, 278 (5706) :748-749
[6]   THIP AND ISOGUVACINE ARE PARTIAL AGONISTS OF GABA-STIMULATED BENZODIAZEPINE RECEPTOR-BINDING [J].
KAROBATH, M ;
LIPPITSCH, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 58 (04) :485-488
[7]   STIMULATION OF BENZODIAZEPINE RECEPTOR-BINDING BY GAMMA-AMINOBUTYRIC ACID [J].
KAROBATH, M ;
SPERK, G .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (02) :1004-1006
[8]   PIPERIDINE-4-SULFONIC ACID - NEW SPECIFIC GABA AGONIST [J].
KROGSGAARDLARSEN, P ;
FALCH, E ;
SCHOUSBOE, A ;
CURTIS, DR ;
LODGE, D .
JOURNAL OF NEUROCHEMISTRY, 1980, 34 (03) :756-759
[9]   NEW CLASS OF GABA AGONIST [J].
KROGSGAARDLARSEN, P ;
JOHNSTON, GAR ;
LODGE, D ;
CURTIS, DR .
NATURE, 1977, 268 (5615) :53-55
[10]   STRUCTURE AND BIOLOGICAL-ACTIVITY OF A SERIES OF CONFORMATIONALLY RESTRICTED ANALOGUES OF GABA [J].
KROGSGAARDLARSEN, P ;
JOHNSTON, GAR ;
CURTIS, DR ;
GAME, CJA ;
MCCULLOCH, RM .
JOURNAL OF NEUROCHEMISTRY, 1975, 25 (06) :803-809