CHARACTERIZATION OF PLATELET THROMBOXANE-A2 PROSTAGLANDIN-H-2 RECEPTOR BY A NOVEL THROMBOXANE RECEPTOR ANTAGONIST, [H-3]S-145

被引:48
作者
HANASAKI, K [1 ]
NAGASAKI, T [1 ]
ARITA, H [1 ]
机构
[1] SHIONOGI & CO LTD, SHIONOGI RES LAB, FUKUSHIMA KU, OSAKA 553, JAPAN
关键词
D O I
10.1016/0006-2952(89)90501-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2007 / 2017
页数:11
相关论文
共 39 条
[1]   LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].
ARMSTRONG, RA ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964
[2]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[3]   HYDRODYNAMIC PROPERTIES OF A THROMBOXANE-A2 PROSTAGLANDIN-H2 ANTAGONIST BINDING-SITE SOLUBILIZED FROM HUMAN-PLATELETS [J].
BURCH, RM ;
MAIS, DE ;
PEPKOWITZ, SH ;
HALUSHKA, PV .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 132 (03) :961-968
[4]   SOLUBILIZATION OF A THROMBOXANE-A2/PROSTAGLANDIN-H2 ANTAGONIST BINDING-SITE FROM HUMAN-PLATELETS [J].
BURCH, RM ;
MAIS, DE ;
SAUSSY, DL ;
HALUSHKA, PV .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (21) :7434-7438
[5]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[6]  
COLEMAN RA, 1980, BRIT J PHARMACOL, V68, pP127
[7]  
DARIUS H, 1985, J PHARMACOL EXP THER, V235, P274
[8]  
DUTTAROY AK, 1987, J BIOL CHEM, V262, P12685
[9]  
HALUSHKA PV, 1987, FASEB J, V46, P131
[10]   THROMBOXANES - NEW GROUP OF BIOLOGICALLY-ACTIVE COMPOUNDS DERIVED FROM PROSTAGLANDIN ENDOPEROXIDES [J].
HAMBERG, M ;
SVENSSON, J ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1975, 72 (08) :2994-2998