SYNTHESIS OF AND GLYCOSIDASE INHIBITION BY ALPHA-L-HOMOFUCONOJIRIMYCIN

被引：21

作者：

ANDREWS, DM

BIRD, MI

CUNNINGHAM, MM

WARD, P

机构：

[1] Glaxo Group Research, Greenford, Middlesex UB6 0HE, Greenford Road

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1993年 / 3卷 / 12期

关键词：

D O I：

10.1016/S0960-894X(01)80711-3

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The first synthesis of the novel azasugar alpha-L-homofuconojirimycin is reported. The biological activity of this compound is described and is shown to be mom specific for alpha-L-fucosidase than compounds previously tested.

引用

页码：2533 / 2536

页数：4

共 7 条

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