RO 18-5364, A POTENT NEW INHIBITOR OF THE GASTRIC (H+ + K+)-ATPASE

被引:15
作者
SIGRISTNELSON, K
KRASSO, A
MULLER, RKM
FISCHLI, AE
机构
[1] F HOFFMANN LA ROCHE & CO LTD, PHARMACEUT RES DEPT, GRENZACHERSTR 124, CH-4002 BASEL, SWITZERLAND
[2] UNIV BERN, DEPT BIOCHEM, CH-3000 BERN, SWITZERLAND
来源
EUROPEAN JOURNAL OF BIOCHEMISTRY | 1987年 / 166卷 / 02期
关键词
D O I
10.1111/j.1432-1033.1987.tb13537.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:453 / 459
页数:7
相关论文
共 20 条
[1]   INHIBITION OF PARTIALLY PURIFIED K+/H+-ATPASE FROM GUINEA-PIG ISOLATED AND ENRICHED PARIETAL-CELLS BY SUBSTITUTED BENZIMIDAZOLES [J].
BEIL, W ;
SEWING, KF .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 82 (03) :651-657
[2]  
FALLER LD, 1985, ENZYMES BIOL MEMBR, V3, P431
[3]   SUBSTITUTED BENZIMIDAZOLES INHIBIT GASTRIC-ACID SECRETION BY BLOCKING (H++K+)ATPASE [J].
FELLENIUS, E ;
BERGLINDH, T ;
SACHS, G ;
OLBE, L ;
ELANDER, B ;
SJOSTRAND, SE ;
WALLMARK, B .
NATURE, 1981, 290 (5802) :159-161
[4]  
Fiske CH, 1925, J BIOL CHEM, V66, P375
[5]   MECHANISMS OF GASTRIC H+ AND CL- TRANSPORT [J].
FORTE, JG ;
MACHEN, TE ;
OBRINK, KJ .
ANNUAL REVIEW OF PHYSIOLOGY, 1980, 42 :111-126
[6]   K+-STIMULATED PHOSPHATASE OF MICROSOMES FROM GASTRIC MUCOSA [J].
FORTE, JG ;
FORTE, GM ;
SALTMAN, P .
JOURNAL OF CELLULAR PHYSIOLOGY, 1967, 69 (03) :293-+
[7]   CORRELATION OF PARIETAL-CELL STRUCTURE AND FUNCTION [J].
FORTE, JG ;
FORTE, TM ;
BLACK, JA ;
OKAMOTO, C ;
WOLOSIN, JM .
JOURNAL OF CLINICAL GASTROENTEROLOGY, 1983, 5 :17-27
[8]  
IM WB, 1985, J BIOL CHEM, V260, P9452
[9]   THE 1ST PRACTICAL METHOD FOR ASYMMETRIC EPOXIDATION [J].
KATSUKI, T ;
SHARPLESS, KB .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (18) :5974-5976
[10]   CLEAVAGE OF STRUCTURAL PROTEINS DURING ASSEMBLY OF HEAD OF BACTERIOPHAGE-T4 [J].
LAEMMLI, UK .
NATURE, 1970, 227 (5259) :680-+