FACILE SYNTHESIS OF 6,7-DICHLORO-1-OXO-5-INDANYLALKANOIC ACIDS AND RELATED COMPOUNDS VIA TRIFLATE DISPLACEMENT

被引：8

作者：

WILLIAMS, HWR ^{[1
]}

ROONEY, CS ^{[1
]}

BICKING, JB ^{[1
]}

ROBB, CM ^{[1
]}

DESOLMS, SJ ^{[1
]}

WOLTERSDORF, OW ^{[1
]}

CRAGOE, EJ ^{[1
]}

机构：

[1] MERCK SHARP & DOHME,RES LABS,W POINT,PA 19486

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1979年 / 44卷 / 23期

关键词：

D O I：

10.1021/jo01337a008

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Substitution of the triflate group in 6, 7-dichloro-l-oxo-5-indanyl trifluoromethanesulfonates, by a conjugative addition-displacement mechanism, provides a new route to 1-indanones with a variety of substituents in the 5-position. © 1979, American Chemical Society. All rights reserved.

引用

页码：4060 / 4063

页数：4

共 7 条

[1]

ATKINSON JG, TETRAHEDRON LETT

[2]

Bayles R., 1977, SYNTHESIS-STUTTGART, V31, P33

[3]

CAVAZZA M, 1977, SYNTHESIS-STUTTGART, P298

[4] DISPLACEMENT OF METHOXY BY AMINO-GROUPS IN ARYLOXAZOLINES - NOVEL-APPROACH TO ORTHO-AMINOBENZOIC, ORTHO-ALKYLAMINOBENZOIC, AND ORTHO-DIALKYLAMINOBENZOIC ACIDS [J].