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SPECIES-DIFFERENCES IN ANTICOAGULANT AND ANTI-XA ACTIVITY OF DX-9065A, A HIGHLY SELECTIVE FACTOR XA INHIBITOR
被引:73
作者
:
HARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories II, Daiichi Pharmaceutical Co., Ltd. Tokyo
HARA, T
YOKOYAMA, A
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories II, Daiichi Pharmaceutical Co., Ltd. Tokyo
YOKOYAMA, A
MORISHIMA, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories II, Daiichi Pharmaceutical Co., Ltd. Tokyo
MORISHIMA, Y
KUNITADA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories II, Daiichi Pharmaceutical Co., Ltd. Tokyo
KUNITADA, S
机构
:
[1]
Exploratory Research Laboratories II, Daiichi Pharmaceutical Co., Ltd. Tokyo
来源
:
THROMBOSIS RESEARCH
|
1995年
/ 80卷
/ 01期
关键词
:
DX-9065A;
SELECTIVE FXA INHIBITOR;
SPECIES DIFFERENCE;
ANTICOAGULANT ACTIVITY;
ANTI-XA ACTIVITY;
NAPAP;
D O I
:
10.1016/0049-3848(95)00155-K
中图分类号
:
R5 [内科学];
学科分类号
:
1002
[临床医学]
;
100201
[内科学]
;
摘要
:
[No abstract available]
引用
收藏
页码:99 / 104
页数:6
相关论文
共 13 条
[1]
THE DETERMINATION OF ENZYME INHIBITOR CONSTANTS
[J].
DIXON, M
论文数:
0
引用数:
0
h-index:
0
DIXON, M
.
BIOCHEMICAL JOURNAL,
1953,
55
(01)
:170
-171
[2]
BOVINE FACTOR X1 (STUART FACTOR) - PRIMARY STRUCTURE OF LIGHT CHAIN
[J].
论文数:
引用数:
h-index:
机构:
ENFIELD, DL
;
论文数:
引用数:
h-index:
机构:
ERICSSON, LH
;
论文数:
引用数:
h-index:
机构:
WALSH, KA
;
论文数:
引用数:
h-index:
机构:
NEURATH, H
;
TITANI, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
TITANI, K
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1975,
72
(01)
:16
-19
[3]
HARA T, 1994, THROMB HAEMOSTASIS, V71, P314
[4]
HARA T, IN PRESS THROMB HAEM
[5]
A NOVEL FACTOR XA INHIBITOR - STRUCTURE-ACTIVITY-RELATIONSHIPS AND SELECTIVITY BETWEEN FACTOR XA AND THROMBIN
[J].
KATAKURA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
KATAKURA, S
;
NAGAHARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
NAGAHARA, T
;
HARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
HARA, T
;
IWAMOTO, M
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
IWAMOTO, M
.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1993,
197
(02)
:965
-972
[6]
GLU-192-]GLN SUBSTITUTION IN THROMBIN MIMICS THE CATALYTIC SWITCH INDUCED BY THROMBOMODULIN
[J].
LEBONNIEC, BF
论文数:
0
引用数:
0
h-index:
0
机构:
OKLAHOMA MED RES FDN,CARDIOVASC BIOL RES PROGRAM,OKLAHOMA CITY,OK 73104
LEBONNIEC, BF
;
ESMON, CT
论文数:
0
引用数:
0
h-index:
0
机构:
OKLAHOMA MED RES FDN,CARDIOVASC BIOL RES PROGRAM,OKLAHOMA CITY,OK 73104
ESMON, CT
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1991,
88
(16)
:7371
-7375
[7]
GENE FOR HUMAN FACTOR-X - A BLOOD-COAGULATION FACTOR WHOSE GENE ORGANIZATION IS ESSENTIALLY IDENTICAL WITH THAT OF FACTOR-IX AND PROTEIN-C
[J].
LEYTUS, SP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
LEYTUS, SP
;
论文数:
引用数:
h-index:
机构:
FOSTER, DC
;
KURACHI, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
KURACHI, K
;
论文数:
引用数:
h-index:
机构:
DAVIE, EW
.
BIOCHEMISTRY,
1986,
25
(18)
:5098
-5102
[8]
THE SYNTHESIS OF SULFATED DEXTRAN BEADS FOR ISOLATION OF HUMAN-PLASMA COAGULATION FACTOR-II, FACTOR-IX, AND FACTOR-X
[J].
MILETICH, JP
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
MILETICH, JP
;
BROZE, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
BROZE, GJ
;
论文数:
引用数:
h-index:
机构:
MAJERUS, PW
.
ANALYTICAL BIOCHEMISTRY,
1980,
105
(02)
:304
-310
[9]
DIBASIC (AMIDINOARYL)PROPANOIC ACID-DERIVATIVES AS NOVEL BLOOD-COAGULATION FACTOR XA INHIBITORS
[J].
NAGAHARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
NAGAHARA, T
;
YOKOYAMA, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
YOKOYAMA, Y
;
INAMURA, K
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
INAMURA, K
;
KATAKURA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
KATAKURA, S
;
KOMORIYA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
KOMORIYA, S
;
YAMAGUCHI, H
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
YAMAGUCHI, H
;
HARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
HARA, T
;
IWAMOTO, M
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
IWAMOTO, M
.
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(08)
:1200
-1207
[10]
PURIFICATION AND CHARACTERIZATION OF RECOMBINANT ANTISTASIN - A LEECH-DERIVED INHIBITOR OF COAGULATION FACTOR-XA
[J].
NUTT, EM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
NUTT, EM
;
JAIN, D
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
JAIN, D
;
LENNY, AB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
LENNY, AB
;
SCHAFFER, L
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
SCHAFFER, L
;
SIEGL, PK
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
SIEGL, PK
;
DUNWIDDIE, CT
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
DUNWIDDIE, CT
.
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1991,
285
(01)
:37
-44
←
1
2
→
共 13 条
[1]
THE DETERMINATION OF ENZYME INHIBITOR CONSTANTS
[J].
DIXON, M
论文数:
0
引用数:
0
h-index:
0
DIXON, M
.
BIOCHEMICAL JOURNAL,
1953,
55
(01)
:170
-171
[2]
BOVINE FACTOR X1 (STUART FACTOR) - PRIMARY STRUCTURE OF LIGHT CHAIN
[J].
论文数:
引用数:
h-index:
机构:
ENFIELD, DL
;
论文数:
引用数:
h-index:
机构:
ERICSSON, LH
;
论文数:
引用数:
h-index:
机构:
WALSH, KA
;
论文数:
引用数:
h-index:
机构:
NEURATH, H
;
TITANI, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
TITANI, K
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1975,
72
(01)
:16
-19
[3]
HARA T, 1994, THROMB HAEMOSTASIS, V71, P314
[4]
HARA T, IN PRESS THROMB HAEM
[5]
A NOVEL FACTOR XA INHIBITOR - STRUCTURE-ACTIVITY-RELATIONSHIPS AND SELECTIVITY BETWEEN FACTOR XA AND THROMBIN
[J].
KATAKURA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
KATAKURA, S
;
NAGAHARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
NAGAHARA, T
;
HARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
HARA, T
;
IWAMOTO, M
论文数:
0
引用数:
0
h-index:
0
机构:
Exploratory Research Laboratories 2, Daiichi Pharmaceutical Co. Ltd., Tokyo 134, 1-16-13 Kita-Kasai, Edogawa-ku
IWAMOTO, M
.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1993,
197
(02)
:965
-972
[6]
GLU-192-]GLN SUBSTITUTION IN THROMBIN MIMICS THE CATALYTIC SWITCH INDUCED BY THROMBOMODULIN
[J].
LEBONNIEC, BF
论文数:
0
引用数:
0
h-index:
0
机构:
OKLAHOMA MED RES FDN,CARDIOVASC BIOL RES PROGRAM,OKLAHOMA CITY,OK 73104
LEBONNIEC, BF
;
ESMON, CT
论文数:
0
引用数:
0
h-index:
0
机构:
OKLAHOMA MED RES FDN,CARDIOVASC BIOL RES PROGRAM,OKLAHOMA CITY,OK 73104
ESMON, CT
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1991,
88
(16)
:7371
-7375
[7]
GENE FOR HUMAN FACTOR-X - A BLOOD-COAGULATION FACTOR WHOSE GENE ORGANIZATION IS ESSENTIALLY IDENTICAL WITH THAT OF FACTOR-IX AND PROTEIN-C
[J].
LEYTUS, SP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
LEYTUS, SP
;
论文数:
引用数:
h-index:
机构:
FOSTER, DC
;
KURACHI, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
UNIV WASHINGTON,DEPT BIOCHEM,SEATTLE,WA 98195
KURACHI, K
;
论文数:
引用数:
h-index:
机构:
DAVIE, EW
.
BIOCHEMISTRY,
1986,
25
(18)
:5098
-5102
[8]
THE SYNTHESIS OF SULFATED DEXTRAN BEADS FOR ISOLATION OF HUMAN-PLASMA COAGULATION FACTOR-II, FACTOR-IX, AND FACTOR-X
[J].
MILETICH, JP
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
MILETICH, JP
;
BROZE, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT BIOL CHEM,DIV HEMATOL ONCOL,ST LOUIS,MO 63110
BROZE, GJ
;
论文数:
引用数:
h-index:
机构:
MAJERUS, PW
.
ANALYTICAL BIOCHEMISTRY,
1980,
105
(02)
:304
-310
[9]
DIBASIC (AMIDINOARYL)PROPANOIC ACID-DERIVATIVES AS NOVEL BLOOD-COAGULATION FACTOR XA INHIBITORS
[J].
NAGAHARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
NAGAHARA, T
;
YOKOYAMA, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
YOKOYAMA, Y
;
INAMURA, K
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
INAMURA, K
;
KATAKURA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
KATAKURA, S
;
KOMORIYA, S
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
KOMORIYA, S
;
YAMAGUCHI, H
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
YAMAGUCHI, H
;
HARA, T
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
HARA, T
;
IWAMOTO, M
论文数:
0
引用数:
0
h-index:
0
机构:
Research Institute, Daiichi Pharmaceutical Company, Ltd., Tokyo 134
IWAMOTO, M
.
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(08)
:1200
-1207
[10]
PURIFICATION AND CHARACTERIZATION OF RECOMBINANT ANTISTASIN - A LEECH-DERIVED INHIBITOR OF COAGULATION FACTOR-XA
[J].
NUTT, EM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
NUTT, EM
;
JAIN, D
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
JAIN, D
;
LENNY, AB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
LENNY, AB
;
SCHAFFER, L
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
SCHAFFER, L
;
SIEGL, PK
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
SIEGL, PK
;
DUNWIDDIE, CT
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME LTD,DEPT BIOL CHEM WP26-431,W POINT,PA 19486
DUNWIDDIE, CT
.
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1991,
285
(01)
:37
-44
←
1
2
→