SUPER-ACTIVE ENKEPHALIN ANALOGS - SIMPLE TRIPEPTIDE HYDROXYALKYLAMIDES EXHIBIT SURPRISINGLY HIGH AND LONG-LASTING OPIOID ACTIVITIES

被引：21

作者：

KISO, Y ^{[1
]}

YAMAGUCHI, M ^{[1
]}

AKITA, T ^{[1
]}

MORITOKI, H ^{[1
]}

TAKEI, M ^{[1
]}

NAKAMURA, H ^{[1
]}

机构：

[1] DAINIPPON PHARMACEUT CO LTD,RES LABS,SUITA,OSAKA 564,JAPAN

来源：

NATURWISSENSCHAFTEN | 1981年 / 68卷 / 04期

关键词：

D O I：

10.1007/BF01047210

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：210 / 212

页数：3

共 26 条

[1] ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT
BELLUZZI, JD
GRANT, N
GARSKY, V
SARANTAKIS, D
WISE, CD
STEIN, L
[J]. NATURE, 1976, 260 (5552) : 625 - 626
[2] EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE
BUSCHER, HH
HILL, RC
ROMER, D
CARDINAUX, F
CLOSSE, A
HAUSER, D
PLESS, J
[J]. NATURE, 1976, 261 (5559) : 423 - 425
[3] D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
[4] EXTREMELY RAPID DEGRADATION OF [H-3] METHIONINE-ENKEPHALIN BY VARIOUS RAT TISSUES INVIVO AND INVITRO
DUPONT, A
CUSAN, L
GARON, M
ALVARADOURBINA, G
LABRIE, F
[J]. LIFE SCIENCES, 1977, 21 (07) : 907 - 914
[5] EDDY NB, 1953, J PHARMACOL EXP THER, V107, P385
[6] TETRAPEPTIDE ACYL-HYDRAZIDE ANALOGS OF ENKEPHALIN - NEW GROUP OF POTENT ANALGESICS
FUJINO, M
SHINAGAWA, S
KAWAI, K
ISHII, H
[J]. NATURWISSENSCHAFTEN, 1979, 66 (12) : 625 - 626
[7] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY
HUGHES, J
SMITH, TW
KOSTERLITZ, HW
FOTHERGILL, LA
MORGAN, BA
MORRIS, HR
[J]. NATURE, 1975, 258 (5536) : 577 - 579
[8] DEPROTECTION OF O-METHYLTYROSINE BY A PUSH-PULL MECHANISM USING THE THIOANISOLE-TRIFLUOROMETHANESULPHONIC ACID SYSTEM - APPLICATION TO THE CONVENIENT SYNTHESIS OF A POTENT N-METHYLENKEPHALIN DERIVATIVE
KISO, Y
NAKAMURA, S
ITO, K
UKAWA, K
KITAGAWA, K
AKITA, T
MORITOKI, H
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1979, (21) : 971 - 972
[9] EFFICIENT REMOVAL OF N-BENZYLOXYCARBONYL GROUP BY A PUSH-PULL MECHANISM USING THIOANISOLE-TRIFLUOROACETIC ACID, EXEMPLIFIED BY A SYNTHESIS OF MET-ENKEPHALIN
KISO, Y
UKAWA, K
AKITA, T
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1980, (03) : 101 - 102
[10] KISO Y, 1980, CHEM PHARM BULL, V28, P673

← 1 2 3 →