A LOW DISTRIBUTION VOLUME AS A DETERMINANT OF EFFICACY AND SAFETY FOR HISTAMINE (H-1) ANTAGONISTS

被引:30
作者
TILLEMENT, JP
机构
[1] Department of Pharmacology, Faculty of Medicine, University of Paris Xii
关键词
D O I
10.1111/j.1398-9995.1995.tb04258.x
中图分类号
R392 [医学免疫学];
学科分类号
100102 ;
摘要
Tillement J‐P. A low distribution volume as a determinant of efficacy and safety for histamine (H1) antagonists. Copyright © 1995, Wiley Blackwell. All rights reserved
引用
收藏
页码:12 / 16
页数:5
相关论文
共 17 条
[1]  
BALTES EL, 1987, CETIRIZINE S P NEW E, P45
[2]   EVIDENCE FOR ISOXICAM BINDING TO SITE-I AS A PRIMARY SITE AND TO SITE-II AS A SECONDARY SITE OF HUMAN-SERUM ALBUMIN [J].
BREE, F ;
NGUYEN, P ;
ALBENGRES, E ;
URIEN, S ;
RIANT, P ;
WELLING, PG ;
TILLEMENT, JP .
BIOCHEMICAL PHARMACOLOGY, 1989, 38 (05) :753-758
[3]  
CHESNE C, 1993, ADV EXP MED BIOL, V331, P113
[4]   CARDIOTOXIC EFFECT WITH CONVULSIONS IN TERFENADINE OVERDOSE [J].
DAVIES, AJ ;
HARINDRA, V ;
MCEWAN, A ;
GHOSE, RR .
BRITISH MEDICAL JOURNAL, 1989, 298 (6669) :325-325
[5]   HISTAMINE-RECEPTORS - SUBCLASSES AND SPECIFIC LIGANDS [J].
HAAKSMA, EEJ ;
LEURS, R ;
TIMMERMAN, H .
PHARMACOLOGY & THERAPEUTICS, 1990, 47 (01) :73-104
[6]  
MATZKE GR, 1987, ANN ALLERGY, V59, P25
[7]   INVIVO BINDING-PROPERTIES OF NONSEDATING ANTIHISTAMINES TO CNS HISTAMINE-RECEPTORS [J].
MCQUADE, RD ;
RICHLAN, K ;
DUFFY, RA ;
CHIPKIN, RE ;
BARNETT, A .
DRUG DEVELOPMENT RESEARCH, 1990, 20 (03) :301-306
[8]   THE PHARMACOLOGY AND MECHANISMS OF ACTION OF HISTAMINE-H1-ANTAGONISTS [J].
RIMMER, SJ ;
CHURCH, MK .
CLINICAL AND EXPERIMENTAL ALLERGY, 1990, 20 :3-17
[9]  
SALE ME, 1993, J ALLERGY CLIN IMMUN, V91, P258
[10]  
Simons F E, 1991, Clin Pharmacokinet, V21, P372