A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED 1H-INDOLES

被引：11

作者：

PRASHAD, M

LAVECCHIA, L

PRASAD, K

REPIC, O

机构：

[1] Chemical Research & Development, Technical R & D, Sandoz Research Institute, Sandoz Pharmaceutical Corporation, East Hanover

[2] Kilo Lab, Sandoz Pharma Ltd.

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 01期

关键词：

D O I：

10.1080/00397919508010793

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A convenient synthesis of 3-substituted IH-indoles via functionalization of enamines, which serve as intermediates in the Leimgruber-Batcho approach, followed by reductive cyclization is described.

引用

页码：95 / 100

页数：6

共 10 条

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