DESIGN OF ANTIANDROGENS AND THEIR MECHANISMS OF ACTION - A CASE-STUDY (ANANDRON)

被引:9
作者
RAYNAUD, JP
FIET, J
LEGOFF, JM
MARTIN, PM
MOGUILEWSKY, M
OJASOO, T
机构
[1] FAC MED NORD, CNRS, UA 1175, MARSEILLE, FRANCE
[2] HOP ST LOUIS, F-75475 PARIS 10, FRANCE
关键词
D O I
10.1159/000180948
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:230 / 241
页数:12
相关论文
共 77 条
[1]   SPECIFIC BINDING OF [METHYLTRIENOLONE-H-3 TO BOTH PROGESTIN AND ANDROGEN BINDING-COMPONENTS IN HUMAN BENIGN PROSTATIC HYPERTROPHY (BPH) [J].
ASSELIN, J ;
MELANCON, R ;
GOURDEAU, Y ;
LABRIE, F ;
BONNE, C ;
RAYNAUD, JP .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1979, 10 (05) :483-486
[3]  
BAILEY M, 1985, BR J PHARM S, V54, pP127
[4]  
BEATTIE CW, 1985, CANCER RES, V45, P4206
[5]  
BELAND G, 1987, PROSTATE CANCER A, V234, P391
[6]   PLASMA-LEVELS OF STEROID GLUCURONIDES IN PREPUBERTAL, ADULT AND ELDERLY MEN [J].
BELANGER, A ;
BROCHU, M ;
CLICHE, J .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1986, 24 (05) :1069-1072
[7]   LEVELS OF PLASMA STEROID GLUCURONIDES IN INTACT AND CASTRATED MEN WITH PROSTATIC-CANCER [J].
BELANGER, A ;
BROCHU, M ;
CLICHE, J .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1986, 62 (05) :812-815
[8]   ASSAY OF ANDROGEN BINDING-SITES BY EXCHANGE WITH METHYLTRIENOLONE (R 1881) [J].
BONNE, C ;
RAYNAUD, JP .
STEROIDS, 1976, 27 (04) :497-507
[9]   ANDROGEN RECEPTOR IN HUMAN-SKIN [J].
BONNE, C ;
SAURAT, JH ;
CHIVOT, M ;
LEHUCHET, D ;
RAYNAUD, JP .
BRITISH JOURNAL OF DERMATOLOGY, 1977, 97 (05) :501-503
[10]  
Brisset J M, 1987, Prog Clin Biol Res, V243A, P411