COMPARATIVE ANTICHOLINERGIC POTENCIES OF R-DISOPYRAMIDE AND S-DISOPYRAMIDE IN LONGITUDINAL MUSCLE STRIPS FROM GUINEA-PIG ILEUM

被引:35
作者
GIACOMINI, KM [1 ]
COX, BM [1 ]
BLASCHKE, TF [1 ]
机构
[1] ADDICT RES FDN,PALO ALTO,CA
关键词
D O I
10.1016/0024-3205(80)90471-3
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1191 / 1197
页数:7
相关论文
共 8 条
[1]  
BURKE TR, J MED CHEM
[2]   MORPHINE-TOLERANT LONGITUDINAL MUSCLE STRIP FROM GUINEA-PIG ILEUM [J].
GOLDSTEIN, A ;
SCHULZ, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1973, 48 (04) :655-666
[3]   DISOPYRAMIDE - REVIEW OF ITS PHARMACOLOGICAL PROPERTIES AND THERAPEUTIC USE IN TREATING CARDIAC-ARRHYTHMIAS [J].
HEEL, RC ;
BROGDEN, RN ;
SPEIGHT, TM ;
AVERY, GS .
DRUGS, 1978, 15 (05) :331-368
[4]   ROLE OF CONCENTRATION-DEPENDENT PLASMA-PROTEIN BINDING IN DISOPYRAMIDE DISPOSITION [J].
MEFFIN, PJ ;
ROBERT, EW ;
WINKLE, RA ;
HARAPAT, S ;
PETERS, FA ;
HARRISON, DC .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (01) :29-46
[5]   ORIGIN OF ACETYLCHOLINE RELEASED FROM GUINEA-PIG INTESTINE AND LONGITUDINAL MUSCLE STRIPS [J].
PATON, WDM ;
ZAR, MA .
JOURNAL OF PHYSIOLOGY-LONDON, 1968, 194 (01) :13-&
[6]   CONGESTIVE HEART-FAILURE CAUSED BY ORAL DISOPYRAMIDE [J].
PODRID, PJ ;
SCHOENEBERGER, A ;
LOWN, B .
NEW ENGLAND JOURNAL OF MEDICINE, 1980, 302 (11) :614-617
[7]   PA, A NEW SCALE FOR THE MEASUREMENT OF DRUG ANTAGONISM [J].
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1947, 2 (03) :189-206
[8]   PA2 AND RECEPTOR DIFFERENTIATION - STATISTICAL-ANALYSIS OF COMPETITIVE ANTAGONISM [J].
TALLARIDA, RJ ;
COWAN, A ;
ADLER, MW .
LIFE SCIENCES, 1979, 25 (08) :637-654