THE USE OF INTERACTION KINETICS TO DISTINGUISH POTENTIAL ANTAGONISTS FROM AGONISTS

被引：25

作者：

RAYNAUD, JP ^{[1
]}

BOUTON, MM ^{[1
]}

OJASOO, T ^{[1
]}

机构：

[1] ROUSSEL UCLAF RES CTR,DEPT BIOCHEM,F-75007 PARIS,FRANCE

来源：

TRENDS IN PHARMACOLOGICAL SCIENCES | 1980年 / 1卷 / 12期

关键词：

D O I：

10.1016/0165-6147(80)90036-X

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：324 / 327

页数：4

共 13 条

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[2] RELEVANCE OF KINETIC-PARAMETERS IN DETERMINATION OF SPECIFIC BINDING TO ESTROGEN-RECEPTOR [J].

BOUTON, MM ;

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[3]

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[4] NUCLEAR BINDING AND RETENTION OF RECEPTOR ESTROGEN COMPLEX - RELATION TO AGONISTIC AND ANTAGONISTIC PROPERTIES OF ESTRIOL [J].

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PECK, EJ .

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[5]

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[6]

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[7] STEROID-HORMONE RECEPTORS AND PHARMACOLOGY [J].

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BOUTON, MM ;

MOGUILEWSKY, M ;

OJASOO, T ;

PHILIBERT, D ;

BECK, G ;

LABRIE, F ;

MORNON, JP .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1980, 12 (JAN) :143-157

[8] ACTION OF A NON-STEROID ANTI-ANDROGEN, RU-23908, IN PERIPHERAL AND CENTRAL TISSUES [J].

RAYNAUD, JP ;

BONNE, C ;

BOUTON, MM ;

LAGACE, L ;

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[9]

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[10]

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