CORRELATION OF ADENOSINE RECEPTOR AFFINITIES AND CARDIOVASCULAR ACTIVITY

被引:52
作者
HAMILTON, HW [1 ]
TAYLOR, MD [1 ]
STEFFEN, RP [1 ]
HALEEN, SJ [1 ]
BRUNS, RF [1 ]
机构
[1] WARNER LAMBERT PARKE DAVIS,PHARMACEUT RES,DEPT PHARMACOL,ANN ARBOR,MI 48105
关键词
D O I
10.1016/0024-3205(87)90542-X
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2295 / 2302
页数:8
相关论文
共 12 条
[1]   ADENOSINE RECEPTORS IN BRAIN MEMBRANES - BINDING OF N6-CYCLOHEXYL[H-3]ADENOSINE AND 1,3-DIETHYL-8-[H-3]PHENYLXANTHINE [J].
BRUNS, RF ;
DALY, JW ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (09) :5547-5551
[2]  
BRUNS RF, 1986, MOL PHARMACOL, V29, P331
[3]   ADENOSINE RELAXES THE AORTA BY INTERACTING WITH AN A2-RECEPTOR AND AN INTRACELLULAR SITE [J].
COLLIS, MG ;
BROWN, CM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 96 (1-2) :61-69
[4]   ADENOSINE-ANALOGS MEDIATING DEPRESSANT EFFECTS ON SYNAPTIC TRANSMISSION IN RAT HIPPOCAMPUS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR THE N6 SUBREGION [J].
DUNWIDDIE, TV ;
WORTH, TS ;
OLSSON, RA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 334 (01) :77-85
[5]   ADENOSINE RECEPTORS MEDIATING CARDIAC DEPRESSION [J].
EVANS, DB ;
SCHENDEN, JA ;
BRISTOL, JA .
LIFE SCIENCES, 1982, 31 (22) :2425-2432
[6]  
Haleen S J, 1985, Life Sci, V36, P127, DOI 10.1016/0024-3205(85)90091-8
[7]   PD-116,948, A HIGHLY SELECTIVE-A1 ADENOSINE RECEPTOR ANTAGONIST [J].
HALEEN, SJ ;
STEFFEN, RP ;
HAMILTON, HW .
LIFE SCIENCES, 1987, 40 (06) :555-561
[8]   NOMENCLATURE OF ADENOSINE RECEPTORS [J].
HAMPRECHT, B ;
VANCALKER, D .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1985, 6 (04) :153-154
[9]  
KUSACHI S, 1983, J PHARMACOL EXP THER, V227, P316
[10]   AN INVESTIGATION OF THE RECEPTORS INVOLVED IN THE CORONARY VASODILATORY EFFECT OF ADENOSINE-ANALOGS [J].
LEUNG, E ;
JOHNSTON, CI ;
WOODCOCK, EA .
CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY, 1985, 12 (05) :515-519