SYNTHESIS OF OPTICALLY-ACTIVE AMIDES FROM BETA-FURYL AND BETA-PHENYL ESTERS BY WAY OF ENZYMATIC AMINOLYSIS

被引：34

作者：

GOTOR, V ^{[1
]}

MENENDEZ, E ^{[1
]}

MOULOUNGUI, Z ^{[1
]}

GASET, A ^{[1
]}

机构：

[1] INPT,ECOLE NATL SUPER CHIM TOULOUSE,CHIM AGROIND LAB,F-31077 TOULOUSE,FRANCE

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1993年 / 20期

关键词：

D O I：

10.1039/p19930002453

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Candida antarctica lipase efficiently catalyses the aminolysis of non-activated esters with a beta-furyl or beta-phenyl group; use of racemic amines gives the corresponding optically active amides with high enantiomeric excess.

引用

页码：2453 / 2456

页数：4

共 9 条

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