CRYSTAL-STRUCTURE STUDIES AND INHIBITION-KINETICS OF TRIPEPTIDE CHLOROMETHYL KETONE INHIBITORS WITH STREPTOMYCES-GRISEUS PROTEASE-B

被引：44

作者：

JAMES, MNG ^{[1
]}

BRAYER, GD ^{[1
]}

DELBAERE, LTJ ^{[1
]}

SIELECKI, AR ^{[1
]}

GERTLER, A ^{[1
]}

机构：

[1] HEBREW UNIV JERUSALEM,JERUSALEM 91000,ISRAEL

来源：

JOURNAL OF MOLECULAR BIOLOGY | 1980年 / 139卷 / 03期

关键词：

D O I：

10.1016/0022-2836(80)90139-4

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：423 / 438

页数：16

共 48 条

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[6] MOLECULAR-STRUCTURE OF CRYSTALLINE STREPTOMYCES-GRISEUS PROTEASE-A AT 2.8-A RESOLUTION .2. MOLECULAR-CONFORMATION, COMPARISON WITH ALPHA-CHYMOTRYPSIN AND ACTIVE-SITE GEOMETRY
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[J]. JOURNAL OF MOLECULAR BIOLOGY, 1978, 124 (01) : 261 - 283
[7] CRYSTALLOGRAPHIC AND KINETIC INVESTIGATIONS OF THE COVALENT COMPLEX FORMED BY A SPECIFIC TETRAPEPTIDE ALDEHYDE AND THE SERINE PROTEASE FROM STREPTOMYCES-GRISEUS
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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (01) : 96 - 100
[8] MOLECULAR-STRUCTURE OF CRYSTALLINE STREPTOMYCES-GRISEUS PROTEASE-A AT 2.8-A RESOLUTION .1. CRYSTALLIZATION, DATA-COLLECTION AND STRUCTURAL-ANALYSIS
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[J]. JOURNAL OF MOLECULAR BIOLOGY, 1978, 124 (01) : 243 - 259
[9] 4.5 A RESOLUTION STRUCTURE OF A BACTERIAL SERINE PROTEASE FROM STREPTOMYCES-GRISEUS
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[J]. CANADIAN JOURNAL OF BIOCHEMISTRY, 1974, 52 (03): : 208 - 220
[10] TERTIARY STRUCTURAL DIFFERENCES BETWEEN MICROBIAL SERINE PROTEASES AND PANCREATIC SERINE ENZYMES
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[J]. NATURE, 1975, 257 (5529) : 758 - 763

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