A GENERAL, CONVENIENT WAY TO CARBORANE-CONTAINING AMINO-ACIDS FOR BORON NEUTRON-CAPTURE THERAPY

被引：46

作者：

WYZLIC, IM

SOLOWAY, AH

机构：

[1] College of Pharmacy, The Ohio State University, Columbus, OH 43210

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 49期

关键词：

D O I：

10.1016/S0040-4039(00)60803-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A general, convenient procedure for the synthesis of carborane-containing amino acids in good yield has been developed. The synthesis of o-carboranylalanine 1, O-(o-carboran-1-ylmethyl)-tyrosine 2 and p-(o-carboran-1-yl)-phenylalanine 3 is reported.

引用

页码：7489 / 7490

页数：2

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