ENHANCEMENT OF MORPHINE ANALGESIA AFTER ACUTE AND CHRONIC HALOPERIDOL

被引:14
作者
HEAD, M
LAL, H
PURI, S
MANTIONE, C
VALENTINO, D
机构
[1] Department of Pharmacology, Toxicology University of Rhode Island, Kingston
关键词
D O I
10.1016/0024-3205(79)90076-6
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
In the male rats haloperidol pretreatment caused an enhancement of morphine analgesia. After chronic haloperidol the analgesia enhancing effect of haloperidol was observed up to 10 days after its discontinuation. No analgesia was present in the haloperidol treated rats not given morphine. © 1979.
引用
收藏
页码:2037 / 2043
页数:7
相关论文
共 28 条
[1]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[2]  
CAVENAR JO, 1976, PSYCHOSOMATICS, V17, P128
[3]   HALOPERIDOL BINDING TO AN OPIATE RECEPTOR-SITE [J].
CLAY, GA ;
BROUGHAM, LR .
BIOCHEMICAL PHARMACOLOGY, 1975, 24 (13-1) :1363-1367
[4]   BUTYROPHENONE INFLUENCES ON OPIATE RECEPTOR [J].
CREESE, I ;
FEINBERG, AP ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1976, 36 (01) :231-235
[5]   H-3-SPIROPERIDOL LABELS DOPAMINE RECEPTORS IN PITUITARY AND BRAIN [J].
CREESE, I ;
SCHNEIDER, R ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 46 (04) :377-381
[6]   HALOPERIDOL-INDUCED TOLERANCE TO MORPHINE CATALEPSY [J].
EZRINWATERS, C ;
SEEMAN, P .
LIFE SCIENCES, 1977, 21 (03) :419-422
[7]  
Fielding S., 1978, HDB PSYCHOPHARMACOLO, VVolume 10, P91
[8]  
GARCIA DA, 1975, LAB ANIM SCI, V25, P585
[9]   ALTERATION IN ACTION OF CHOLINERGIC AND ANTICHOLINERGIC DRUGS AFTER CHRONIC HALOPERIDOL - INDIRECT EVIDENCE FOR CHOLINERGIC HYPOSENSITIVITY [J].
GIANUTSOS, G ;
LAL, H .
LIFE SCIENCES, 1976, 18 (05) :515-520
[10]  
HONG JS, 1978, J PHARMACOL EXP THER, V205, P141