TISSUE SELECTIVITY OF THE CHOLESTEROL-LOWERING AGENTS LOVASTATIN, SIMVASTATIN AND PRAVASTATIN IN RATS INVIVO

被引:158
作者
GERMERSHAUSEN, JI
HUNT, VM
BOSTEDOR, RG
BAILEY, PJ
KARKAS, JD
ALBERTS, AW
机构
关键词
D O I
10.1016/0006-291X(89)92773-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:667 / 675
页数:9
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共 12 条
  • [1] MEVINOLIN - A HIGHLY POTENT COMPETITIVE INHIBITOR OF HYDROXYMETHYLGLUTARYL-COENZYME-A REDUCTASE AND A CHOLESTEROL-LOWERING AGENT
    ALBERTS, AW
    CHEN, J
    KURON, G
    HUNT, V
    HUFF, J
    HOFFMAN, C
    ROTHROCK, J
    LOPEZ, M
    JOSHUA, H
    HARRIS, E
    PATCHETT, A
    MONAGHAN, R
    CURRIE, S
    STAPLEY, E
    ALBERSSCHONBERG, G
    HENSENS, O
    HIRSHFIELD, J
    HOOGSTEEN, K
    LIESCH, J
    SPRINGER, J
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (07): : 3957 - 3961
  • [2] BROWN AG, 1976, J CHEM SOC PERK T, V1, P1165
  • [3] MONACOLIN-K, A NEW HYPOCHOLESTEROLEMIC AGENT PRODUCED BY A MONASCUS SPECIES
    ENDO, A
    [J]. JOURNAL OF ANTIBIOTICS, 1979, 32 (08) : 852 - 854
  • [4] ML-236A, ML-236B, AND ML-236C, NEW INHIBITORS OF CHOLESTEROGENESIS PRODUCED BY PENICILLIUM CITRINUM
    ENDO, A
    KURODA, M
    TSUJITA, Y
    [J]. JOURNAL OF ANTIBIOTICS, 1976, 29 (12) : 1346 - 1348
  • [5] HARUYAMA H, 1986, CHEM PHARM BULL, V34, P1459
  • [6] HELLER RA, 1976, J BIOL CHEM, V251, P3815
  • [7] HOFFMAN WF, 1986, J MED CHEM, V29, P849, DOI 10.1021/jm00155a040
  • [8] PURIFICATION OF 3-HYDROXY-3-METHYLGLUTARYL-COENZYME-A REDUCTASE FROM RAT-LIVER
    KLEINSEK, DA
    RANGANATHAN, S
    PORTER, JW
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (04) : 1431 - 1435
  • [9] MICROBIAL HYDROXYLATION OF ML-236B (COMPACTIN) - STUDIES ON MICROORGANISMS CAPABLE OF 3-BETA-HYDROXYLATION OF ML-236B
    SERIZAWA, N
    SERIZAWA, S
    NAKAGAWA, K
    FURUYA, K
    OKAZAKI, T
    TERAHARA, A
    [J]. JOURNAL OF ANTIBIOTICS, 1983, 36 (07) : 887 - 891