SYNERGISM BETWEEN 9-DEAZAINOSINE AND DL-ALPHA-DIFLUOROMETHYLORNITHINE IN TREATMENT OF EXPERIMENTAL AFRICAN TRYPANOSOMIASIS

被引:29
作者
BACCHI, CJ
BERENS, RL
NATHAN, HC
KLEIN, RS
ELEGBE, IA
RAO, KVB
MCCANN, PP
MARR, JJ
机构
[1] PACE UNIV,DEPT BIOL,NEW YORK,NY 10038
[2] UNIV COLORADO,HLTH SCI CTR,DIV INFECT DIS,DENVER,CO 80262
[3] MEM SLOAN KETTERING CANC CTR,SLOAN KETTERING INST CANC RES,ORGAN CHEM LAB,NEW YORK,NY 10021
[4] MERRELL DOW PHARMACEUT INC,RES INST,CINCINNATI,OH 45215
关键词
D O I
10.1128/AAC.31.9.1406
中图分类号
Q93 [微生物学];
学科分类号
071005 ; 100705 ;
摘要
引用
收藏
页码:1406 / 1413
页数:8
相关论文
共 38 条
[1]  
Bacchi C.J., 1987, P317
[2]   POLYAMINE METABOLISM - A POTENTIAL THERAPEUTIC TARGET IN TRYPANOSOMES [J].
BACCHI, CJ ;
NATHAN, HC ;
HUTNER, SH .
SCIENCE, 1980, 210 (4467) :332-334
[3]   INVIVO EFFECTS OF ALPHA-DL-DIFLUOROMETHYLORNITHINE ON THE METABOLISM AND MORPHOLOGY OF TRYPANOSOMA-BRUCEI-BRUCEI [J].
BACCHI, CJ ;
GAROFALO, J ;
MOCKENHAUPT, D ;
MCCANN, PP ;
DIEKEMA, KA ;
PEGG, AE ;
NATHAN, HC ;
MULLANEY, EA ;
CHUNOSOFF, L ;
SJOERDSMA, A ;
HUTNER, SH .
MOLECULAR AND BIOCHEMICAL PARASITOLOGY, 1983, 7 (03) :209-225
[4]  
BACCHI CJ, 1987, AM J TROP MED HYG, V36, P48
[5]   PYRAZOLOPYRIMIDINE METABOLISM IN AFRICAN TRYPANOSOMES - METABOLIC SIMILARITIES TO TRYPANOSOMA-CRUZI AND LEISHMANIA SPP [J].
BERENS, RL ;
MARR, JJ ;
BRUN, R .
MOLECULAR AND BIOCHEMICAL PARASITOLOGY, 1980, 1 (02) :69-73
[6]   METABOLISM OF FORMYCIN-B BY LEISHMANIA AMASTIGOTES INVITRO - COMPARATIVE METABOLISM IN INFECTED AND UNINFECTED HUMAN MACROPHAGES [J].
BERMAN, JD ;
RAINEY, P ;
SANTI, DV .
JOURNAL OF EXPERIMENTAL MEDICINE, 1983, 158 (01) :252-257
[7]   ACTIVITY OF PURINE ANALOGS AGAINST LEISHMANIA-DONOVANI INVIVO [J].
BERMAN, JD ;
HANSON, WL ;
LOVELACE, JK ;
WAITS, VB ;
JACKSON, JE ;
CHAPMAN, WL ;
KLEIN, RS .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1987, 31 (01) :111-113
[8]   ACTIVITY OF PURINE ANALOGS AGAINST LEISHMANIA-TROPICA WITHIN HUMAN MACROPHAGES INVITRO [J].
BERMAN, JD ;
LEE, LS ;
ROBINS, RK ;
REVANKAR, GR .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1983, 24 (02) :233-236
[9]   CATALYTIC IRREVERSIBLE INHIBITION OF TRYPANOSOMA-BRUCEI-BRUCEI ORNITHINE DECARBOXYLASE BY SUBSTRATE AND PRODUCT ANALOGS AND THEIR EFFECTS ON MURINE TRYPANOSOMIASIS [J].
BITONTI, AJ ;
BACCHI, CJ ;
MCCANN, PP ;
SJOERDSMA, A .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (10) :1773-1777
[10]   PHOSPHORYLATION AND ANTI-LEISHMANIAL ACTIVITY OF FORMYCIN-B [J].
CARSON, DA ;
CHANG, KP .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 100 (03) :1377-1383