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ALPHA-ADRENOCEPTORS AND BETA-ADRENOCEPTORS - FROM THE GENE TO THE CLINIC .2. STRUCTURE-ACTIVITY-RELATIONSHIPS AND THERAPEUTIC APPLICATIONS
被引:197
作者
:
RUFFOLO, RR
论文数:
0
引用数:
0
h-index:
0
机构:
Division of Pharmacological Sciences, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406-0939
RUFFOLO, RR
BONDINELL, W
论文数:
0
引用数:
0
h-index:
0
机构:
Division of Pharmacological Sciences, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406-0939
BONDINELL, W
HIEBLE, JP
论文数:
0
引用数:
0
h-index:
0
机构:
Division of Pharmacological Sciences, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406-0939
HIEBLE, JP
机构
:
[1]
Division of Pharmacological Sciences, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406-0939
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1995年
/ 38卷
/ 19期
关键词
:
D O I
:
10.1021/jm00019a001
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
[No abstract available]
引用
收藏
页码:3681 / 3716
页数:36
相关论文
共 318 条
[1]
ABOUMOHAMED G, 1994, J CARDIOVASC PHARM, V23, P492
[2]
AGHAJANIAN GK, 1985, PSYCHIAT LETT, V111, P57
[3]
AHO M, 1992, ANESTH ANALG, V75, P932
[4]
AHO M, 1992, ANESTH ANALG, V75, P940
[5]
ALPHA-2-ADRENOCEPTOR BLOCKING PROFILE OF SK-AND-F-104078 - FURTHER EVIDENCE FOR RECEPTOR SUBTYPES
AKERS, I
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
AKERS, I
COATES, J
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
COATES, J
DREW, GM
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
DREW, GM
SULLIVAN, AT
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
SULLIVAN, AT
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1991,
102
(04)
: 943
-
949
[6]
BW-A575C, A CHEMICALLY NOVEL AGENT WITH ANGIOTENSIN CONVERTING-ENZYME-INHIBITOR AND BETA-ADRENOCEPTOR-BLOCKING PROPERTIES
ALLAN, G
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
ALLAN, G
CAMBRIDGE, D
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
CAMBRIDGE, D
HARDY, GW
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
HARDY, GW
FOLLENFANT, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
FOLLENFANT, MJ
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1987,
90
(03)
: 609
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615
[7]
INVIVO PHARMACOLOGICAL PROFILE OF SL-84.0418, A NEW SELECTIVE, PERIPHERALLY ACTIVE ALPHA-2-ADRENOCEPTOR ANTAGONIST
ANGEL, I
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
ANGEL, I
GROSSET, A
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
GROSSET, A
PERRAULT, G
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
PERRAULT, G
SHOEMAKER, H
论文数:
0
引用数:
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h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
SHOEMAKER, H
LANGER, SZ
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h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
LANGER, SZ
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1993,
234
(2-3)
: 137
-
145
[8]
ANGEL I, 1992, J PHARMACOL EXP THER, V263, P137
[9]
ATYPICAL BETA-ADRENOCEPTOR ON BROWN ADIPOCYTES AS TARGET FOR ANTI-OBESITY DRUGS
ARCH, JRS
论文数:
0
引用数:
0
h-index:
0
ARCH, JRS
AINSWORTH, AT
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0
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0
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0
AINSWORTH, AT
CAWTHORNE, MA
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PIERCY, V
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SENNITT, MV
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THODY, VE
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WILSON, S
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0
引用数:
0
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WILSON, S
[J].
NATURE,
1984,
309
(5964)
: 163
-
165
[10]
ELECTROPHYSIOLOGIC ACTIVITY AND ANTIARRHYTHMIC EFFICACY OF CK-3579, A NEW CLASS-III ANTIARRHYTHMIC AGENT WITH BETA-ADRENERGIC BLOCKING PROPERTIES
ARGENTIERI, TM
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
ARGENTIERI, TM
TROY, HH
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
TROY, HH
CARROLL, MS
论文数:
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引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
CARROLL, MS
DOROSHUK, CM
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
DOROSHUK, CM
SULLIVAN, ME
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
SULLIVAN, ME
[J].
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1993,
21
(04)
: 647
-
655
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共 318 条
[1]
ABOUMOHAMED G, 1994, J CARDIOVASC PHARM, V23, P492
[2]
AGHAJANIAN GK, 1985, PSYCHIAT LETT, V111, P57
[3]
AHO M, 1992, ANESTH ANALG, V75, P932
[4]
AHO M, 1992, ANESTH ANALG, V75, P940
[5]
ALPHA-2-ADRENOCEPTOR BLOCKING PROFILE OF SK-AND-F-104078 - FURTHER EVIDENCE FOR RECEPTOR SUBTYPES
AKERS, I
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
AKERS, I
COATES, J
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
COATES, J
DREW, GM
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
DREW, GM
SULLIVAN, AT
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
GLAXO GRP RES LTD,DEPT GASTROINTESTINAL PHARMACOL,WARE SG12 0DP,HERTS,ENGLAND
SULLIVAN, AT
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1991,
102
(04)
: 943
-
949
[6]
BW-A575C, A CHEMICALLY NOVEL AGENT WITH ANGIOTENSIN CONVERTING-ENZYME-INHIBITOR AND BETA-ADRENOCEPTOR-BLOCKING PROPERTIES
ALLAN, G
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
ALLAN, G
CAMBRIDGE, D
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
CAMBRIDGE, D
HARDY, GW
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
HARDY, GW
FOLLENFANT, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND
FOLLENFANT, MJ
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1987,
90
(03)
: 609
-
615
[7]
INVIVO PHARMACOLOGICAL PROFILE OF SL-84.0418, A NEW SELECTIVE, PERIPHERALLY ACTIVE ALPHA-2-ADRENOCEPTOR ANTAGONIST
ANGEL, I
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
ANGEL, I
GROSSET, A
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
GROSSET, A
PERRAULT, G
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
PERRAULT, G
SHOEMAKER, H
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
SHOEMAKER, H
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
DEPT BIOL,SYNTHELABO RECH,LERS,31 AVE PAUL VAILLANT COUTURIER,BP 110,F-92225 BAGNEUX,FRANCE
LANGER, SZ
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1993,
234
(2-3)
: 137
-
145
[8]
ANGEL I, 1992, J PHARMACOL EXP THER, V263, P137
[9]
ATYPICAL BETA-ADRENOCEPTOR ON BROWN ADIPOCYTES AS TARGET FOR ANTI-OBESITY DRUGS
ARCH, JRS
论文数:
0
引用数:
0
h-index:
0
ARCH, JRS
AINSWORTH, AT
论文数:
0
引用数:
0
h-index:
0
AINSWORTH, AT
CAWTHORNE, MA
论文数:
0
引用数:
0
h-index:
0
CAWTHORNE, MA
PIERCY, V
论文数:
0
引用数:
0
h-index:
0
PIERCY, V
SENNITT, MV
论文数:
0
引用数:
0
h-index:
0
SENNITT, MV
THODY, VE
论文数:
0
引用数:
0
h-index:
0
THODY, VE
WILSON, C
论文数:
0
引用数:
0
h-index:
0
WILSON, C
WILSON, S
论文数:
0
引用数:
0
h-index:
0
WILSON, S
[J].
NATURE,
1984,
309
(5964)
: 163
-
165
[10]
ELECTROPHYSIOLOGIC ACTIVITY AND ANTIARRHYTHMIC EFFICACY OF CK-3579, A NEW CLASS-III ANTIARRHYTHMIC AGENT WITH BETA-ADRENERGIC BLOCKING PROPERTIES
ARGENTIERI, TM
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
ARGENTIERI, TM
TROY, HH
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
TROY, HH
CARROLL, MS
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
CARROLL, MS
DOROSHUK, CM
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
DOROSHUK, CM
SULLIVAN, ME
论文数:
0
引用数:
0
h-index:
0
机构:
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
BERLEX LABS INC, DEPT BIOL RES, CEDAR KNOLLS, NJ USA
SULLIVAN, ME
[J].
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1993,
21
(04)
: 647
-
655
←
1
2
3
4
5
6
7
8
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→