ALPHA-ADRENOCEPTORS AND BETA-ADRENOCEPTORS - FROM THE GENE TO THE CLINIC .2. STRUCTURE-ACTIVITY-RELATIONSHIPS AND THERAPEUTIC APPLICATIONS

被引:197
作者
RUFFOLO, RR
BONDINELL, W
HIEBLE, JP
机构
[1] Division of Pharmacological Sciences, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406-0939
关键词
D O I
10.1021/jm00019a001
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:3681 / 3716
页数:36
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共 318 条
  • [1] ABOUMOHAMED G, 1994, J CARDIOVASC PHARM, V23, P492
  • [2] AGHAJANIAN GK, 1985, PSYCHIAT LETT, V111, P57
  • [3] AHO M, 1992, ANESTH ANALG, V75, P932
  • [4] AHO M, 1992, ANESTH ANALG, V75, P940
  • [5] ALPHA-2-ADRENOCEPTOR BLOCKING PROFILE OF SK-AND-F-104078 - FURTHER EVIDENCE FOR RECEPTOR SUBTYPES
    AKERS, I
    COATES, J
    DREW, GM
    SULLIVAN, AT
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1991, 102 (04) : 943 - 949
  • [6] BW-A575C, A CHEMICALLY NOVEL AGENT WITH ANGIOTENSIN CONVERTING-ENZYME-INHIBITOR AND BETA-ADRENOCEPTOR-BLOCKING PROPERTIES
    ALLAN, G
    CAMBRIDGE, D
    HARDY, GW
    FOLLENFANT, MJ
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1987, 90 (03) : 609 - 615
  • [7] INVIVO PHARMACOLOGICAL PROFILE OF SL-84.0418, A NEW SELECTIVE, PERIPHERALLY ACTIVE ALPHA-2-ADRENOCEPTOR ANTAGONIST
    ANGEL, I
    GROSSET, A
    PERRAULT, G
    SHOEMAKER, H
    LANGER, SZ
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1993, 234 (2-3) : 137 - 145
  • [8] ANGEL I, 1992, J PHARMACOL EXP THER, V263, P137
  • [9] ATYPICAL BETA-ADRENOCEPTOR ON BROWN ADIPOCYTES AS TARGET FOR ANTI-OBESITY DRUGS
    ARCH, JRS
    AINSWORTH, AT
    CAWTHORNE, MA
    PIERCY, V
    SENNITT, MV
    THODY, VE
    WILSON, C
    WILSON, S
    [J]. NATURE, 1984, 309 (5964) : 163 - 165
  • [10] ELECTROPHYSIOLOGIC ACTIVITY AND ANTIARRHYTHMIC EFFICACY OF CK-3579, A NEW CLASS-III ANTIARRHYTHMIC AGENT WITH BETA-ADRENERGIC BLOCKING PROPERTIES
    ARGENTIERI, TM
    TROY, HH
    CARROLL, MS
    DOROSHUK, CM
    SULLIVAN, ME
    [J]. JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 21 (04) : 647 - 655