SYNTHESIS AND PRELIMINARY PHARMACOLOGICAL EVALUATION OF ASYMMETRIC CHLOROQUINE ANALOGS

被引：8

作者：

WITIAK, DT ^{[1
]}

GRATTAN, DA ^{[1
]}

HEASLIP, RJ ^{[1
]}

RAHWAN, RG ^{[1
]}

机构：

[1] OHIO STATE UNIV,COLL PHARM,DEPT PHARMACOL,COLUMBUS,OH 43210

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 06期

关键词：

D O I：

10.1021/jm00138a014

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：712 / 717

页数：6

共 26 条

[1]

AKESSON CE, 1980, RES COMMUN CHEM PATH, V27, P265

[2]

Bennett MR., 1972, AUTONOMIC NEUROMUSCU

[3]

DAY RA, 1974, QUANTITATIVE ANAL, P145

[4] INHIBITING EFFECTS OF MORPHINE, CHLOROQUINE, NONSTEROIDAL AND STEROIDAL ANTI-INFLAMMATORY DRUGS ON ELECTRICALLY-INDUCED CONTRACTIONS OF GUINEA-PIG ILEUM AND REVERSING EFFECT OF PROSTAGLANDINS [J].

FAMAEY, JP ;

FONTAINE, J ;

REUSE, J .

AGENTS AND ACTIONS, 1975, 5 (04) :354-358

[5] ANALYSIS OF INHIBITORY EFFECTS AND OF POSSIBLE PROSTAGLANDINS ANTAGONISM OF CHLOROQUINE IN GUINEA-PIG ISOLATED ILEUM [J].

FAMAEY, JP ;

FONTAINE, J ;

REUSE, J .

JOURNAL OF PHARMACY AND PHARMACOLOGY, 1977, 29 (12) :761-762

[6]

GREENBERG S, 1973, ARCH INT PHARMACOD T, V205, P381

[7]

GRZONKA Z, 1974, SYNTHESIS-STUTTGART, P661

[8]

HABERKORN A, 1979, TROPENMED PARASITOL, V30, P308

[9] ASPIRIN, INDOMETHACIN, CATECHOLAMINE AND PROSTAGLANDIN INTERACTIONS ON RAT ARTERIOLES AND RABBIT HEARTS [J].

HORROBIN, DF ;

MANKU, MS ;

KARMALI, R ;

NASSAR, BA ;

DAVIES, PA .

NATURE, 1974, 250 (5465) :425-426

[10] CHLOROQUINE, QUININE, PROCAINE, QUINIDINE AND CLOMIPRAMINE ARE PROSTAGLANDIN AGONISTS AND ANTAGONISTS [J].

MANKU, MS ;

HORROBIN, DF .

PROSTAGLANDINS, 1976, 12 (05) :789-801

← 1 2 3 →