PHACLOFEN ANTAGONIZES GABA AT AUTORECEPTORS REGULATING RELEASE IN RAT CEREBRAL-CORTEX

被引:27
作者
BONANNO, G [1 ]
FONTANA, G [1 ]
RAITERI, M [1 ]
机构
[1] UNIV GENOVA,IST FARMACOL & FARMACOGNOSIA,VIALE CEMBRANO 4,I-16148 GENOVA,ITALY
关键词
D O I
10.1016/0014-2999(88)90104-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:223 / 224
页数:2
相关论文
共 5 条
  • [1] A PHYSIOLOGICAL-ROLE FOR GABAB RECEPTORS IN THE CENTRAL NERVOUS-SYSTEM
    DUTAR, P
    NICOLL, RA
    [J]. NATURE, 1988, 332 (6160) : 156 - 158
  • [2] BACLOFEN-H-3 AND H-3-GABA BIND TO BICUCULLINE-INSENSITIVE GABA-B SITES IN RAT-BRAIN
    HILL, DR
    BOWERY, NG
    [J]. NATURE, 1981, 290 (5802) : 149 - 152
  • [3] PHACLOFEN - A PERIPHERAL AND CENTRAL BACLOFEN ANTAGONIST
    KERR, DIB
    ONG, J
    PRAGER, RH
    GYNTHER, BD
    CURTIS, DR
    [J]. BRAIN RESEARCH, 1987, 405 (01) : 150 - 154
  • [4] STUDIES ON [H-3] GABA AND ENDOGENOUS GABA RELEASE IN RAT CEREBRAL-CORTEX SUGGEST THE PRESENCE OF AUTORECEPTORS OF THE GABA-B TYPE
    PITTALUGA, A
    ASARO, D
    PELLEGRINI, G
    RAITERI, M
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 144 (01) : 45 - 52
  • [5] RAITERI M, 1978, REV NEUROSCI-SERIES, V3, P77