A POTENT RADIOLABELED HUMAN RENIN INHIBITOR, [H-3] SR42128 - ENZYMATIC, KINETIC, AND BINDING-STUDIES TO RENIN AND OTHER ASPARTIC PROTEASES

被引：9

作者：

CUMIN, F

NISATO, D

GAGNOL, JP

CORVOL, P

机构：

[1] INSERM,U3617,F-75005 PARIS,FRANCE

[2] SANOFI RECH,F-34082 MONTPELLIER,FRANCE

来源：

BIOCHEMISTRY | 1987年 / 26卷 / 24期

关键词：

D O I：

10.1021/bi00398a013

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：7615 / 7621

页数：7

共 30 条

[1] 3-DIMENSIONAL STRUCTURE, SPECIFICITY AND CATALYTIC MECHANISM OF RENIN
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PEARL, L
[J]. NATURE, 1983, 304 (5923) : 273 - 275
[2] NOVEL RENIN INHIBITORS CONTAINING THE AMINO-ACID STATINE
BOGER, J
LOHR, NS
ULM, EH
POE, M
BLAINE, EH
FANELLI, GM
LIN, TY
PAYNE, LS
SCHORN, TW
LAMONT, BI
VASSIL, TC
STABILITO, II
VEBER, DF
RICH, DH
BOPARI, AS
[J]. NATURE, 1983, 303 (5912) : 81 - 84
[3] RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE
BOGER, J
PAYNE, LS
PERLOW, DS
LOHR, NS
POE, M
BLAINE, EH
ULM, EH
SCHORN, TW
LAMONT, BI
LIN, TY
KAWAI, M
RICH, DH
VEBER, DF
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) : 1779 - 1790
[4] 3-DIMENSIONAL STRUCTURE OF THE COMPLEX OF THE RHIZOPUS-CHINENSIS CARBOXYL PROTEINASE AND PEPSTATIN AT 2.5-A RESOLUTION
BOTT, R
SUBRAMANIAN, E
DAVIES, DR
[J]. BIOCHEMISTRY, 1982, 21 (26) : 6956 - 6962
[5] BREIPOHL G, 1984, THERAPIEWOCHE, V34, P6370
[6] COMPETITIVE INHIBITORS OF RENIN INHIBITORS EFFECTIVE AT PHYSIOLOGICAL PH
BURTON, J
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HABER, E
[J]. BIOCHEMISTRY, 1975, 14 (17) : 3892 - 3898
[7] CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[8] STATISTICAL TEST OF MODELS AND COMPUTERIZED PARAMETER-ESTIMATION FOR ALDOSTERONE BINDING IN RAT-KIDNEY
CLAIRE, M
RAFESTINOBLIN, ME
MICHAUD, A
CORVOL, P
VENOT, A
ROTHMEYER, C
BOISVIEUX, JF
MALLET, A
[J]. FEBS LETTERS, 1978, 88 (02) : 295 - 299
[9] CUMIN F, 1985, J BIOL CHEM, V260, P9154
[10] DECLAVIERE M, 1985, J CARDIOVASC PHAR S4, V7, P558

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