SYNTHESIS, ANTIPARASITIC AND ANTIFUNGAL ACTIVITIES OF ARYLALKYL AND ARYLVINYLTHIAZOLINES

被引：19

作者：

CAUJOLLE, R

BAZIARDMOUYSSET, G

FAVROT, JD

PAYARD, M

LOISEAU, PR

AMAROUCH, H

LINAS, MD

SEGUELA, JP

LOISEAU, PM

BORIES, C

GAYRAL, P

机构：

[1] LAB PARASITOL,F-92290 CHATENAY MALABRY,FRANCE

[2] CHU RANGUEIL,SERV PARASITOL MYCOL,F-31054 TOULOUSE,FRANCE

[3] FAC SCI CASABLANCA,LASABLANCA,MOROCCO

来源：

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1993年 / 28卷 / 01期

关键词：

ANTIPARASITIC; ANTHELMINTIC; ANTIFUNGAL ACTIVITY; ARYLALKYLTHIAZOLINES; ARYLVINYLTHIAZOLINES;

D O I：

10.1016/0223-5234(93)90076-Q

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Twenty-seven arylalkyl- or arylvinylthiazolines were synthesized and tested in vitro against three genera of nematodes, various yeasts and opportunistic fungi. Vinyl compounds seem to have an interesting filaricidal activity against Molinema dessetae and anti-fungal activity against yeasts.

引用

页码：29 / 35

页数：7

共 13 条

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